Organic Letters Home Page (ACS Publications)

ACS Publications: High Quality, High Impact

Brief reports of significant research concerning organic chemistry, including organic synthesis, organometallic, natural product, physical organic, bioorganic, and medicinal chemistry.

Editors: Amos B. Smith, III & Associate Editors

Volume: 10, 24 issues

Division of Organic Chemistry
Division of Medicinal Chemistry

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The Most Recently Published Research

The following list of Articles ASAP is limited to the latest 20 articles. Visit the All Articles ASAP page for the complete listing.

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Web Release Date: July 8, 2008

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Chuktabrins A and B, Two Novel Limonoids from the Twigs and Leaves of Chukrasia tabularis
Chuan-Rui Zhang, Cheng-Qi Fan, Li Zhang, Sheng-Ping Yang, Yan Wu, Yang Lu, and Jian-Min Yue
Web Release Date: 08-Jul-2008; (Letter) DOI: 10.1021/ol800885h

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Web Release Date: July 4, 2008

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Arylation of Phe and Tyr Side Chains of Unprotected Peptides by a Suzuki−Miyaura Reaction in Water
Maria Vilaró, Gemma Arsequell, Gregorio Valencia, Alfredo Ballesteros, and José Barluenga
Web Release Date: 04-Jul-2008; (Letter) DOI: 10.1021/ol801009z

Abstract Full: HTML / PDF (91K) Supporting Info

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Synthesis of 3-Selena-1-dethiacephems and Selenazepines via Iodocyclization
Dinesh R. Garud and Mamoru Koketsu
Web Release Date: 04-Jul-2008; (Letter) DOI: 10.1021/ol801010y

Abstract Full: HTML / PDF (297K) Supporting Info

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Colorimetric Discrimination between Important Alkaloid Nuclei Mediated by a Bis-Salphen Chromophore
Sander J. Wezenberg, Eduardo C. Escudero-Adán, Jordi Benet-Buchholz, and Arjan W. Kleij
Web Release Date: 04-Jul-2008; (Letter) DOI: 10.1021/ol801167r

Abstract Full: HTML / PDF (974K) Supporting Info

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A Regio- and Stereocontrolled Approach to Pyranosyl C-Nucleoside Synthesis
Philip Redpath, Simon Macdonald, and Marie E. Migaud
Web Release Date: 04-Jul-2008; (Letter) DOI: 10.1021/ol801183e

Abstract Full: HTML / PDF (141K) Supporting Info

Web Release Date: July 3, 2008

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Efficient Synthesis of 2-Substituted-1,2,3-triazoles
Jarosław Kalisiak, K. Barry Sharpless, and Valery V. Fokin
Web Release Date: 03-Jul-2008; (Letter) DOI: 10.1021/ol8006748

Abstract Full: HTML / PDF (346K) Supporting Info

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Photochemistry of Allenyl Salicylaldehydes
Frédéric Birbaum, Antonia Neels, and Christian G. Bochet
Web Release Date: 03-Jul-2008; (Letter) DOI: 10.1021/ol800806a

Abstract Full: HTML / PDF (245K) Supporting Info

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Synthetic Studies on (+)-Manzamine A: Stereoselective Synthesis of the Tetracyclic Core Framework
Yoichi Kita, Tatsuya Toma, Toshiyuki Kan, and Tohru Fukuyama
Web Release Date: 03-Jul-2008; (Letter) DOI: 10.1021/ol801111r

Abstract Full: HTML / PDF (120K) Supporting Info

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An Unexpected Phosphine-Catalyzed [3 + 2] Annulation. Synthesis of Highly Functionalized Cyclopentenes
Zheng Lu, Suqing Zheng, Xumu Zhang, and Xiyan Lu
Web Release Date: 03-Jul-2008; (Letter) DOI: 10.1021/ol8011452

Abstract Full: HTML / PDF (129K) Supporting Info

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Iron(II) Bromide-Catalyzed Synthesis of Benzimidazoles from Aryl Azides
Meihua Shen and Tom G. Driver
Web Release Date: 03-Jul-2008; (Letter) DOI: 10.1021/ol801227f

Abstract Full: HTML / PDF (126K) Supporting Info

Web Release Date: July 2, 2008

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Copper-Catalyzed Intramolecular Cyclization to N-Substituted 1,3-Dihydrobenzimidazol-2-ones
Zhaoguang Li, Hongbin Sun, Hualiang Jiang, and Hong Liu
Web Release Date: 02-Jul-2008; (Letter) DOI: 10.1021/ol8011106

Abstract Full: HTML / PDF (109K) Supporting Info

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Efficient and Selective Syntheses of (all-E)- and (6E,10Z)-2′-O-Methylmyxalamides D via Pd-Catalyzed Alkenylation−Carbonyl Olefination Synergy
Guangwei Wang, Zhihong Huang, and Ei-ichi Negishi
Web Release Date: 02-Jul-2008; (Letter) DOI: 10.1021/ol801115s

Abstract Full: HTML / PDF (914K) Supporting Info

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Enantioselective Organocatalytic Formal [3 + 3]-Cycloaddition of α,β-Unsaturated Aldehydes and Application to the Asymmetric Synthesis of (−)-Isopulegol Hydrate and (−)-Cubebaol
Bor-Cherng Hong, Ming-Fun Wu, Hsing-Chang Tseng, and Ju-Hsiou Liao
Web Release Date: 02-Jul-2008; (Additions & Corrections) DOI: 10.1021/ol8014144

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Web Release Date: July 1, 2008

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Solid-Support Based Total Synthesis and Stereochemical Correction of Brunsvicamide A
Thilo Walther, Hans-Dieter Arndt, and Herbert Waldmann
Web Release Date: 01-Jul-2008; (Letter) DOI: 10.1021/ol801064d

Abstract Full: HTML / PDF (764K) Supporting Info

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Synthesis of the (3R,6S)-3-Amino-6-(2,3-difluorophenyl)azepan-2-one of Telcagepant (MK-0974), a Calcitonin Gene-Related Peptide Receptor Antagonist for the Treatment of Migraine Headache
Christopher S. Burgey, Daniel V. Paone, Anthony W. Shaw, James Z. Deng, Diem N. Nguyen, Craig M. Potteiger, Samuel L. Graham, Joseph P. Vacca, and Theresa M. Williams
Web Release Date: 01-Jul-2008; (Letter) DOI: 10.1021/ol8011524

Abstract Full: HTML / PDF (127K) Supporting Info

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Carbonyl Groups as Molecular Valves to Regulate Chloride Binding to Squaramides
Vijayakumar Ramalingam, Maciej E. Domaradzki, Seogjoo Jang, and Rajeev S. Muthyala
Web Release Date: 01-Jul-2008; (Letter) DOI: 10.1021/ol801204s

Abstract Full: HTML / PDF (430K) Supporting Info

Web Release Date: June 28, 2008

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Copper-Catalyzed Sonogashira-Type Reactions Under Mild Palladium-Free Conditions
Florian Monnier, François Turtaut, Leslie Duroure, and Marc Taillefer
Web Release Date: 28-Jun-2008; (Letter) DOI: 10.1021/ol801025u

Abstract Full: HTML / PDF (203K) Supporting Info

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A Panchromatic Boradiazaindacene (BODIPY) Sensitizer for Dye-Sensitized Solar Cells
Sule Erten-Ela, M. Deniz Yilmaz, Burcak Icli, Yavuz Dede, Siddik Icli, and Engin U. Akkaya
Web Release Date: 28-Jun-2008; (Letter) DOI: 10.1021/ol8010612

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Palladium-Catalyzed Hydrophosphorylation and Hydrophosphinylation of Cyclopropenes
Bassam K. Alnasleh, William M. Sherrill, and Michael Rubin
Web Release Date: 28-Jun-2008; (Letter) DOI: 10.1021/ol8011138