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Article

Regiospecific and Stereoselective Syntheses of (±)-Reserpine and (−)-Reserpine

Supporting Info

Gilbert Stork,* Peng Cho Tang,^† Michael Casey,^‡ Burton Goodman,^§ and Masahiro Toyota

Contribution from the Department of Chemistry, Columbia University, New York, New York 10027

J. Am. Chem. Soc., 2005, 127 (46), pp 16255–16262

DOI: 10.1021/ja055744x

Publication Date (Web): November 1, 2005

In papers with more than one author, the asterisk indicates the name of the author to whom inquiries about the paper should be addressed.

†

Hengrui Pharmaceutical Ltd., Shanghai.

‡

University College, Dublin.

Deceased Dec 28, 2004.

Osaka Prefecture University.

, gjs8@columbia.edu

Abstract

Full details of three approaches to an entirely regio- and stereoselective synthesis of the well-known target reserpine are described, culminating in a total synthesis which efficiently meets these requirements.

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Published In Issue November 23, 2005
Received August 22, 2005

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Article

Regiospecific and Stereoselective Syntheses of (±)-Reserpine and (−)-Reserpine

Abstract

Tools

SciFinder Links

History

Recommend & Share

Related Content

Enantiospecific Total Syntheses of Kapakahines B and F

A Short and Efficient Synthesis of (−)-7-Methylomuralide, a Potent Proteasome Inhibitor

Enantioselective Total Synthesis of (−)-Napyradiomycin A1 via Asymmetric Chlorination of an Isolated Olefin

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