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Concise Formation of 4-Benzyl Piperidines and Related Derivatives Using a Suzuki Protocol

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Susan Vice,* Tom Bara, Annette Bauer, C. Anderson Evans, Jennifer Ford, Hubert Josien, Stuart McCombie,* Michael Miller, Dennis Nazareno, Anandan Palani, and Jay Tagat

ScheringPlough Research Institute, 2015 Galloping Hill Road, Kenilworth, New Jersey 07033-0539sfvice@home.com

J. Org. Chem., 2001, 66 (7), pp 2487–2492

DOI: 10.1021/jo0007682

Publication Date (Web): March 3, 2001

To whom correspondence should be addressed. (S.F.V.) Phone: (908)789-1206. Fax: (908)791-1992. E-mail: sfvice@home.com. (S.M.) Schering-Plough Research Institute, 2015 Galloping Hill Rd., Kenilworth, NJ, 07033-0593. Phone: (908)740-3544. Fax: (908)740-7512. E-mail: stuart.mccombie@spcorp.com.

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Published In Issue April 06, 2001
Received May 19, 2000
Revised January 30, 2001

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