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Synthesis of Tertiary Benzamides via Pd-Catalyzed Coupling of Arylboronic Esters and Carbamoyl Chlorides

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Morten Lysén, Susan Kelleher, Mikael Begtrup, and Jesper Langgaard Kristensen*

Department of Medicinal Chemistry, Danish University of Pharmaceutical Sciences, Universitetsparken 2, DK-2100 Copenhagen, Denmark jekr@dfuni.dk

J. Org. Chem., 2005, 70 (13), pp 5342–5343

DOI: 10.1021/jo050459h

Publication Date (Web): May 21, 2005

In papers with more than one author, the asterisk indicates the name of the author to whom inquiries about the paper should be addressed.

Abstract

Ortho-substituted arylboronic esters are efficiently coupled with carbamoyl chlorides under Pd-catalysis to give tertiary benzamides.

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Published In Issue June 24, 2005
Received March 9, 2005

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Note

Synthesis of Tertiary Benzamides via Pd-Catalyzed Coupling of Arylboronic Esters and Carbamoyl Chlorides

Abstract

Tools

SciFinder Links

History

Recommend & Share

Related Content

Total Synthesis of (−)-Penifulvin A, an Insecticide with a Dioxafenestrane Skeleton

Copper(II) Acetate-Catalyzed Addition of Arylboronic Acids to Aromatic Aldehydes

Versatile Pd(II)-Catalyzed C−H Activation/Aryl−Aryl Coupling of Benzoic and Phenyl Acetic Acids

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