Cart
Article
Highly Enantioselective Synthesis of β-Amino Alcohols: A Catalytic Version
Full Text HTML
Hi-Res PDFPurchase the full-text
- PDF/HTML,
figures/images,
references and tables,
(where available)
Section:Abstract
Highly enantioselective rearrangement of β-amino alcohols was realized by using a catalytic amount of trifluoroacetic anhydride.
Citing Articles
Citation data is made available by participants in CrossRef's Cited-by Linking service. For a more comprehensive list of citations to this article, users are encouraged to perform a search in SciFinder.
This article has been cited by 7 ACS Journal articles (5 most recent appear below).
Mild Reaction Conditions for the Terminal Deuteration of Alkynes
Sean P. Bew, Glyn D. Hiatt-Gipson, Jenny. A. Lovell, and Christophe PoullainOrganic Letters2012 14 (2), 456-459Mild Reaction Conditions for the Terminal Deuteration of Alkynes
Sean P. Bew, Glyn D. Hiatt-Gipson, Jenny. A. Lovell, and Christophe PoullainOrganic Letters2012 14 (2), 456-459Routinely employed syntheses of terminally deuterated alkynes often utilize strong bases (i.e., LDA, n-BuLi, or Grignard reagents) or low (i.e., −78 °C) or elevated (i.e., 56 °C) reaction temperatures; furthermore many of these procedures afford average ...
Synthesis of Enantiopure Substituted Piperidines via an Aziridinium Ring Expansion
Scott B. D. Jarvis and Andre B. CharetteOrganic Letters2011 Article ASAPSynthesis of Enantiopure Substituted Piperidines via an Aziridinium Ring Expansion
Scott B. D. Jarvis and Andre B. CharetteOrganic Letters2011 Article ASAPHerein we report a novel methodology for the asymmetric synthesis of 3-substituted piperidines from readily available chiral building blocks. This method, which features a novel irreversible dihydropyrole-tetrahydropyridine ring expansion, allows the ...
One-Pot Stereoselective Synthesis of 1,2-Amino Alcohol Derivatives
Alicia Boto and Iván Romero-EstudilloOrganic Letters2011 Article ASAPOne-Pot Stereoselective Synthesis of 1,2-Amino Alcohol Derivatives
Alicia Boto and Iván Romero-EstudilloOrganic Letters2011 Article ASAPCommon β-hydroxy amino acids (such as threonine) can be readily transformed into 1,2-amino alcohols with excellent stereoselectivity. This one-pot decarboxylation–alkylation process allows the replacement of the carboxyl group by alkyl, allyl, or aryl ...
Asymmetric Synthesis of an Antagonist of Neurokinin Receptors: SSR 241586
Thomas-Xavier Métro, Anne Cochi, Domingo Gomez Pardo, and Janine CossyThe Journal of Organic Chemistry2011 76 (8), 2594-2602Asymmetric Synthesis of an Antagonist of Neurokinin Receptors: SSR 241586
Thomas-Xavier Métro, Anne Cochi, Domingo Gomez Pardo, and Janine CossyThe Journal of Organic Chemistry2011 76 (8), 2594-2602SSR 241586 is a 2,2-disubstituted morpholine, developed by Sanofi-Aventis, which is active in the treatment of schizophrenia and irritable bowel syndrome (IBS). Different strategies have been studied to synthesize this molecule and among the strategies an ...
Assessing the Rates of Ring-Opening of Aziridinium and Azetidinium Ions: A Dramatic Ring Size Effect
Nicolas De Rycke, Olivier David, and François CoutyOrganic Letters2011 13 (7), 1836-1839Assessing the Rates of Ring-Opening of Aziridinium and Azetidinium Ions: A Dramatic Ring Size Effect
Nicolas De Rycke, Olivier David, and François CoutyOrganic Letters2011 13 (7), 1836-1839Rates for the ring-opening of aziridinium and azetidinium ions by DMAP were measured. The four-membered ring appears to be ca. 17 000 times less reactive compared to the three-membered ring but is still highly relevant from a synthetic viewpoint. The ...
Tools
-
Add to Favorites
-
Download Citation
-
Email a Colleague -
Permalink
Order Reprints
Rights & Permissions
Citation Alerts
History
- Published In Issue August 17, 2007
- Received May 16, 2007
ACS
Network
Facebook
Tweet This
CiteULike
Newsvine
Digg This
Delicious
