Boc-Protected Amines via a Mild and Efficient One-Pot Curtius Rearrangement

Related Content

• Diphenylphosphoryl azide. New convenient reagent for a modified Curtius reaction and for peptide synthesisDiphenylphosphoryl azide. New convenient reagent for a modified Curtius reaction and for peptide synthesisJournal of the American Chemical Society

  • Diphenylphosphoryl azide. New convenient reagent for a modified Curtius reaction and for peptide synthesisDiphenylphosphoryl azide. New convenient reagent for a modified Curtius reaction and for peptide synthesis

    Takayuki Shioiri, Kunihiro Ninomiya, Shunichi Yamada
    Journal of the American Chemical Society 1972 94 (17), pp 6203–6205
    Abstract | Hi-Res PDF
• Azides: their preparation and synthetic usesAzides: their preparation and synthetic usesChemical Reviews

  • Azides: their preparation and synthetic usesAzides: their preparation and synthetic uses

    Eric F. V. Scriven, Kenneth Turnbull
    Chemical Reviews 1988 88 (2), pp 297–368
    Abstract | Hi-Res PDF
• An Efficient Synthesis of a Probe for Protein Function:  2,3-Diaminopropionic Acid with Orthogonal Protecting GroupsOrganic Letters

  • An Efficient Synthesis of a Probe for Protein Function:  2,3-Diaminopropionic Acid with Orthogonal Protecting Groups

    Ethan A. Englund, Hosahudya N. Gopi, and Daniel H. Appella
    Organic Letters 2004 6 (2), pp 213–215

    Abstract: An efficient and cost-effective synthesis of N(α)-Boc₂-N(β)-Cbz-2,3-diaminopropionic acid is reported. The synthesis starts from commercially available N(α)-Boc-Asp(OBn)-OH and employs a Curtius rearrangement to establish the β-nitrogen. Proper protection ...

    Abstract | Full Text HTML | Hi-Res PDF

Other ACS content by these authors:

• Hélène Lebel
• Olivier Leogane