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Letter

Direct Pd-Catalyzed Arylation of 1,2,3-Triazoles^†

Stepan Chuprakov, Natalia Chernyak, Alexander S. Dudnik, and Vladimir Gevorgyan*

Department of Chemistry, University of Illinois at Chicago, 845 West Taylor Street, Chicago, Illinois 60607-7061

Org. Lett., 2007, 9 (12), pp 2333–2336

DOI: 10.1021/ol070697u

Publication Date (Web): May 10, 2007

†

Dedicated to Prof. Ivars Kalvins on occasion of his 60th birthday.

In papers with more than one author, the asterisk indicates the name of the author to whom inquiries about the paper should be addressed.

A highly efficient method for the synthesis of multisubstituted 1,2,3-triazoles via a direct Pd-catalyzed C-5 arylation has been developed.

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