Department of Chemistry, Simon Fraser University, Burnaby, British Columbia, Canada, and F. Hoffmann-La Roche AG, pRED, Pharma Research & Early Development, Small Molecule Research, Medicinal Chemistry, Grenzacherstrasse 124, 4070 Basel, Switzerland
A continuous flow inverse-electron-demand Kondrat’eva reaction has been developed that provides direct access to cycloalka[c]pyridines from unactivated oxazoles and cycloalkenes. Annulated pyridines obtained by this one-step process are valuable scaffolds for medicinal chemistry.
Experimental procedures and characterization data for all new compounds. This material is available free of charge via the Internet at http://pubs.acs.org.
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