The Journal of Organic Chemistry: Articles ASAP (ACS Publications)

Facile Syntheses of Enantiopure 3-Hydroxypiperidine Derivatives and 3-Hydroxypipecolic Acids

Wen-Hua Chiou, Gau-Hong Lin and Chih-Wei Liang

Publication Date (Web): February 8, 2010 (Note)

DOI: 10.1021/jo902324h

Regioselective Control in the Oxidative Cleavage of 4,6-O-Benzylidene Acetals of Glycopyranosides by Dimethyldioxirane

Arnaud St

venin, Fran

ois-Didier Boyer and Jean-Marie Beau

Publication Date (Web): February 8, 2010 (Note)

DOI: 10.1021/jo9026098

Palladium-Catalyzed Decarboxylative Cross-Coupling Reaction Between Heteroaromatic Carboxylic Acids and Aryl Halides

Fran

ois Bilodeau, Marie-Christine Brochu, Nicolas Guimond, Kris H. Thesen and Pat Forgione

Publication Date (Web): February 8, 2010 (Article)

DOI: 10.1021/jo9022793

Aqueous Iodine(III)-Mediated Stereoselective Oxidative Cyclization for the Synthesis of Functionalized Fused Dihydrofuran Derivatives

Yang Ye, Linfei Wang and Renhua Fan

Publication Date (Web): February 8, 2010 (Note)

DOI: 10.1021/jo902553k

Synthesis of a Triptycene-Derived Bisparaphenylene-34-crown-10 and Its Complexation with Both Paraquat and Cyclobis(paraquat-p-phenylene)

Yi Jiang, Jing Cao, Jian-Min Zhao, Jun-Feng Xiang and Chuan-Feng Chen

Publication Date (Web): February 8, 2010 (Note)

DOI: 10.1021/jo902571n

Iridium-Catalyzed (Z)-Trialkylsilylation of Terminal Olefins

Biao Lu and J. R. Falck

Publication Date (Web): February 8, 2010 (Article)

DOI: 10.1021/jo902678p

February 5, 2010

Intramolecular Double Proton Transfer from 2-Hydroxy-2-iminoacetic Acid to 2-Amino-2-oxoacetic Acid

Barbara Bankiewicz, Sławomir Wojtulewski and Sławomir J. Grabowski

Publication Date (Web): February 5, 2010 (Article)

DOI: 10.1021/jo9022414

Chiral Bifunctional Thiourea-Catalyzed Enantioselective Michael Addition of Ketones to Nitrodienes

Hai Ma, Kun Liu, Fa-Guang Zhang, Chuan-Le Zhu, Jing Nie and Jun-An Ma

Publication Date (Web): February 5, 2010 (Article)

DOI: 10.1021/jo901991v

Synthesis of Heteroatom Substituted Naphthoporphyrazine Derivatives with Near-Infrared Absorption and Emission

Evan R. Trivedi, Sangwan Lee, Hong Zong, Carl M. Blumenfeld, Anthony G. M. Barrett and Brian M. Hoffman

Publication Date (Web): February 5, 2010 (Note)

DOI: 10.1021/jo9026947

Conformational Analysis of a Model for the trans-Fused FGH Ether Rings in Brevetoxin A

Evan B. Wang and Carol A. Parish

Publication Date (Web): February 5, 2010 (Article)

DOI: 10.1021/jo902558h

February 4, 2010

2-Pyridylnitrene and 3-Pyridazylcarbene and Their Relationship via Ring-Expansion, Ring-Opening, Ring-Contraction, and Fragmentation

David Kvaskoff, Pawel Bednarek and Curt Wentrup

Publication Date (Web): February 4, 2010 (Article)

DOI: 10.1021/jo902570d

Enantioselective Synthesis of α-Quaternary Amino Acid Derivatives by Sequential Enzymatic Desymmetrization and Curtius Rearrangement of α,α-Disubstituted Malonate Diesters

Violeta Iosub, Anton R. Haberl, Jennifer Leung, Michael Tang, Kannan Vembaiyan, Masood Parvez and Thomas G. Back

Publication Date (Web): February 4, 2010 (Article)

DOI: 10.1021/jo902584r

Nucleophilic Catalysis of Carbohydrate Oxime Formation by Anilines

Mikkel B. Thygesen, Henrik Munch, Jørgen Sauer, Emiliano Cl

, Malene R. Jørgensen, Ole Hindsgaul and Knud J. Jensen

Publication Date (Web): February 4, 2010 (Note)

DOI: 10.1021/jo902425v

Enantioselective Carbonyl Allylation, Crotylation, and tert-Prenylation of Furan Methanols and Furfurals via Iridium-Catalyzed Transfer Hydrogenation

Benjamin Bechem, Ryan L. Patman, A. Stephen K. Hashmi and Michael J. Krische

Publication Date (Web): February 4, 2010 (Note)

DOI: 10.1021/jo902697g

Iron(III)-Catalyzed Four-Component Coupling Reaction of 1,3-Dicarbonyl Compounds, Amines, Aldehydes, and Nitroalkanes: A Simple and Direct Synthesis of Functionalized Pyrroles

Sukhendu Maiti, Srijit Biswas and Umasish Jana

Publication Date (Web): February 4, 2010 (Article)

DOI: 10.1021/jo902661y

Domino Heck−Aza-Michael Reactions: Efficient Access to 1-Substituted Tetrahydro-β-carbolines

Daniel L. Priebbenow, Luke C. Henderson, Frederick M. Pfeffer and Scott G. Stewart

Publication Date (Web): February 4, 2010 (Note)

DOI: 10.1021/jo902652h

February 3, 2010

Asymmetric Synthesis of a Potent, Aminopiperidine-Fused Imidazopyridine Dipeptidyl Peptidase IV Inhibitor

Feng Xu, Edward Corley, Michael Zacuto, David A. Conlon, Brenda Pipik, Guy Humphrey, Jerry Murry and David Tschaen

Publication Date (Web): February 3, 2010 (Featured Article)

DOI: 10.1021/jo902573q

Exploring Photoinduced Decarboxylation Mechanism of o-Acetylphenylacetic Acid from the Combined CASSCF and DFT Studies

Lina Ding and Wei-Hai Fang

Publication Date (Web): February 3, 2010 (Article)

DOI: 10.1021/jo902593s

Total Synthesis of (+)-Crocacin C Using Hidden Symmetry

Mathieu Candy, G

rard Audran, Hugues Bienaym

, Cyril Bressy and Jean-Marc Pons

Publication Date (Web): February 3, 2010 (Featured Article)

DOI: 10.1021/jo902582w

Mechanism and Regioselectivity of the Osmium-Catalyzed Aminohydroxylation of Olefins

Dominik Munz and Thomas Strassner

Publication Date (Web): February 3, 2010 (Article)

DOI: 10.1021/jo902421n

Iodine/Palladium Approaches to the Synthesis of Polyheterocyclic Compounds

Saurabh Mehta and Richard C. Larock

Publication Date (Web): February 3, 2010 (Article)

DOI: 10.1021/jo902639f

February 2, 2010

(1R)-(+)-Camphor and Acetone Derived α′-Hydroxy Enones in Asymmetric Diels−Alder Reaction: Catalytic Activation by Lewis and Brønsted Acids, Substrate Scope, Applications in Syntheses, and Mechanistic Studies

Patricia Ba

uelos, Jes

s M. Garc

a, Enrique G

mez-Bengoa, Ada Herrero, Jos

M. Odriozola, Mikel Oiarbide, Claudio Palomo and Jes

s Razkin

Publication Date (Web): February 2, 2010 (Article)

DOI: 10.1021/jo9023039

Scope and Limitations of an Efficient Four-Component Reaction for Dihydropyridin-2-ones

Rachel Scheffelaar, Monica Paravidino, Anass Znabet, Rob F. Schmitz, Frans J. J. de Kanter, Martin Lutz, Anthony L. Spek, C

lia Fonseca Guerra, F. Matthias Bickelhaupt, Marinus B. Groen, Eelco Ruijter and Romano V. A. Orru

Publication Date (Web): February 2, 2010 (Article)

DOI: 10.1021/jo902613j

Reactivity of a Hypervalent Iodine Trifluoromethylating Reagent toward THF: Ring Opening and Formation of Trifluoromethyl Ethers

Serena Fantasia, Jan M. Welch and Antonio Togni

Publication Date (Web): February 2, 2010 (Note)

DOI: 10.1021/jo9025429

Advantageous Use of ^tBu₂P-N═P(ⁱBuNCH₂CH₂)₃N in the Hiyama Coupling of Aryl Bromides and Chlorides

Steven M. Raders, Jesudoss V. Kingston and John G. Verkade

Publication Date (Web): February 2, 2010 (Note)

DOI: 10.1021/jo902338w

February 1, 2010

Dissecting a Dyotropic Rearrangement

Rebecca L. Davis and Dean J. Tantillo

Publication Date (Web): February 1, 2010 (Article)

DOI: 10.1021/jo902685x

Synthesis of ω-Hydroxy Carboxylic Acids and α,ω-Dimethyl Ketones Using α,ω-Diols As Alkylating Agents

Yosuke Iuchi, Megumi Hyotanishi, Brittany E. Miller, Kensaku Maeda, Yasushi Obora and Yasutaka Ishii

Publication Date (Web): February 1, 2010 (Note)

DOI: 10.1021/jo9027165

Reactivity of the Mutagen 1,4-Dinitro-2-methylpyrrole as an Alkylating Agent

M. Teresa P

rez-Prior, Rafael G

mez-Bombarelli, Marina Gonz

lez-P

rez, Jos

A. Manso, M. Pilar Garc

a-Santos, Emilio Calle and Julio Casado

Publication Date (Web): February 1, 2010 (Article)

DOI: 10.1021/jo902329q

An Efficient Preparation of N-Methyl-α-amino Acids from N-Nosyl-α-amino Acid Phenacyl Esters

Antonella Leggio, Emilia Lucia Belsito, Rosaria De Marco, Angelo Liguori, Francesca Perri and Maria Caterina Viscomi

Publication Date (Web): February 1, 2010 (Article)

DOI: 10.1021/jo901643f

De Novo Synthesis of Long-Wavelength Absorbing Chlorin-13,15-dicarboximides

Marcin Ptaszek, Doroth

e Lahaye, Michael Krayer, Chinnasamy Muthiah and Jonathan S. Lindsey

Publication Date (Web): February 1, 2010 (Article)

DOI: 10.1021/jo902649d

Efficient Microwave-Assisted Synthesis of Unsymmetrical Disulfides

Kristina G

rmer, Herbert Waldmann and Gemma Triola

Publication Date (Web): February 1, 2010 (Note)

DOI: 10.1021/jo902695a

January 29, 2010

Effect of Alkyl Substituents on Photorelease from Butyrophenone Derivatives

Sivaramakrishnan Muthukrishnan, Jagadis Sankaranarayanan, Tamara C. S. Pace, Armands Konosonoks, Mariel E. DeMichiei, Michael J. Meese, Cornelia Bohne and Anna D. Gudmundsdottir

Publication Date (Web): January 29, 2010 (Article)

DOI: 10.1021/jo9021088

Stereoselective Synthesis of an Active Metabolite of the Potent PI3 Kinase Inhibitor PKI-179

Zecheng Chen, Aranapakam M. Venkatesan, Osvaldo Dos Santos, Efren Delos Santos, Christoph M. Dehnhardt, Semiramis Ayral-Kaloustian, Joseph Ashcroft, Leonard A. McDonald and Tarek S. Mansour

Publication Date (Web): January 29, 2010 (Article)

DOI: 10.1021/jo9026269

Linear and V-Shaped Nonlinear Optical Chromophores with Multiple 4H-Pyran-4-ylidene Moieties

Raquel Andreu, Elena Gal

n, Javier Gar

n, Vanessa Herrero, Edurne Lacarra, Jes

s Orduna, Raquel Alicante and Bel

n Villacampa

Publication Date (Web): January 29, 2010 (Article)

DOI: 10.1021/jo902670z

Diastereoselective Synthesis of a Highly Functionalized Angularly Substituted cis-Perhydroisoquinoline-3,6-dione via Organoiron

Jeng-Liang Han, Meng-Chi Liu and Chi Wi Ong

Publication Date (Web): January 29, 2010 (Article)

DOI: 10.1021/jo902605w

Sulfoxide-Directed Intramolecular [4 + 2] Cycloadditions between 2-Sulfinyl Butadienes and Unactivated Alkynes

Roberto Fern

ndez de la Pradilla, Mariola Tortosa, Esther Castellanos, Alma Viso and Raquel Baile

Publication Date (Web): January 29, 2010 (Article)

DOI: 10.1021/jo9024489

Synthesis of and Evidence for Electronic Communication within Heteromultimetallic Tetrakis(NCN-pincer metal)−(Metallo)porphyrin Hybrids

Bart M. J. M. Suijkerbuijk, Duncan M. Tooke, Martin Lutz, Anthony L. Spek, Leonardus W. Jenneskens, Gerard van Koten and Robertus J. M. Klein Gebbink

Publication Date (Web): January 29, 2010 (Article)

DOI: 10.1021/jo902402g

Enantioselective Construction of Cis-2,6-Disubstituted Dihydropyrans: Total Synthesis of (−)-Centrolobine

Wojciech Chaładaj, Rafał Kowalczyk and Janusz Jurczak

Publication Date (Web): January 29, 2010 (Note)

DOI: 10.1021/jo902167r

January 28, 2010

A Facile and Efficient Synthesis of 3,3-Dimethyl Isopropylidene Proline From (+)-3-Carene

Latha G. Nair, Anil Saksena, Raymond Lovey, Mousumi Sannigrahi, Jesse Wong, Jianshe Kong, Xiaoyong Fu and Viyyoor Girijavallabhan

Publication Date (Web): January 28, 2010 (Note)

DOI: 10.1021/jo9022759

Asymmetry in the N-Inversion of Heteroarene Imines: Pyrimidin-4(3H)-Imine, Pyridin-2(1H)-Imine, and 1H-Purine-6(9H)-Imine

Rainer Glaser, Jian Yin and Stephanie Miller

Publication Date (Web): January 28, 2010 (Article)

DOI: 10.1021/jo902358c

Erosion of Stereochemical Control with Increasing Nucleophilicity: O-Glycosylation at the Diffusion Limit

Matthew G. Beaver and K. A. Woerpel

Publication Date (Web): January 28, 2010 (Article)

DOI: 10.1021/jo902222a

Zn(OTf)₂-Catalyzed Reactions of Ethenetricarboxylates with 2-Aminobenzaldehydes Leading to Tetrahydroquinoline Derivatives

Shoko Yamazaki, Masachika Takebayashi and Kazuya Miyazaki

Publication Date (Web): January 28, 2010 (Article)

DOI: 10.1021/jo902430v

Superarming Common Glycosyl Donors by Simple 2-O-Benzoyl-3,4,6-tri-O-benzyl Protection

Hemali D. Premathilake, Laurel K. Mydock and Alexei V. Demchenko

Publication Date (Web): January 28, 2010 (Article)

DOI: 10.1021/jo9021474

Solarylations via 4-Aminophenyl Cations

Valentina Dichiarante, Maurizio Fagnoni and Angelo Albini

Publication Date (Web): January 28, 2010 (Article)

DOI: 10.1021/jo902669j

January 27, 2010

PdCl₂(HNMe₂)₂-Catalyzed Highly Selective Cross [2 + 2 + 2] Cyclization of Alkynoates and Alkenes under Molecular Oxygen

Yanxia Shen, Huanfeng Jiang and Zhengwang Chen

Publication Date (Web): January 27, 2010 (Note)

DOI: 10.1021/jo902636g

Large-Scale Asymmetric Synthesis of a Cathepsin S Inhibitor

Jon C. Lorenz, Carl A. Busacca, XuWu Feng, Nelu Grinberg, Nizar Haddad, Joe Johnson, Suresh Kapadia, Heewon Lee, Anjan Saha, Max Sarvestani, Earl M. Spinelli, Rich Varsolona, Xudong Wei, Xingzhong Zeng and Chris H. Senanayake

Publication Date (Web): January 27, 2010 (Article)

DOI: 10.1021/jo9022809

Computational Studies of Ion-Pair Separation of Benzylic Organolithium Compounds in THF: Importance of Explicit and Implicit Solvation

Nipa Deora and Paul R. Carlier

Publication Date (Web): January 27, 2010 (Article)

DOI: 10.1021/jo9016452

January 26, 2010

Au/Ag-Cocatalyzed Aldoximes to Amides Rearrangement under Solvent- and Acid-Free Conditions

Rub

n S. Ram

n, Johann Bosson, Silvia D

ez-Gonz

lez, Nicolas Marion and Steven P. Nolan

Publication Date (Web): January 26, 2010 (Article)

DOI: 10.1021/jo902461a

A Method for the Synthesis of Substituted Quinolines via Electrophilic Cyclization of 1-Azido-2-(2-propynyl)benzene

Zhibao Huo, Ilya D. Gridnev and Yoshinori Yamamoto

Publication Date (Web): January 26, 2010 (Article)

DOI: 10.1021/jo902603v

January 25, 2010

Systematic Investigation of CD Spectra of Aryl Benzyl Sulfoxides Interpreted by Means of TDDFT Calculations

Gennaro Pescitelli, Sebastiano Di Pietro, Cosimo Cardellicchio, Maria Annunziata M. Capozzi and Lorenzo Di Bari

Publication Date (Web): January 25, 2010 (Article)

DOI: 10.1021/jo902363c

Strongly Emitting Fluorophores Based on 1-Azaperylene Scaffold

Daniel T. Gryko, Joanna Piechowska and Michał Gał

zowski

Publication Date (Web): January 25, 2010 (Note)

DOI: 10.1021/jo902443s

Synthesis, Properties, Crystal Structures, and Semiconductor Characteristics of Naphtho[1,2-b:5,6-b′]dithiophene and -diselenophene Derivatives

Shoji Shinamura, Eigo Miyazaki and Kazuo Takimiya

Publication Date (Web): January 25, 2010 (Article)

DOI: 10.1021/jo902545a

A Rapid and Efficient Sonogashira Protocol and Improved Synthesis of Free Fatty Acid 1 (FFA1) Receptor Agonists

Elisabeth Christiansen, Maria E. Due-Hansen and Trond Ulven

Publication Date (Web): January 25, 2010 (Note)

DOI: 10.1021/jo902533p

Enzymatic Deprotection of the Cephalosporin 3′-Acetoxy Group Using Candida antarctica Lipase B

Leslie D. Patterson and Marvin J. Miller

Publication Date (Web): January 25, 2010 (Note)

DOI: 10.1021/jo902406b

Equations for the Transfer of Neutral Molecules and Ionic Species from Water to Organic phases

Michael H Abraham and William E Acree, Jr.

Publication Date (Web): January 25, 2010 (Featured Article)

DOI: 10.1021/jo902388n

January 22, 2010

Preparation of a Storable Zinc Carbenoid Species and Its Application in Cyclopropanation, Chain Extension, and [2,3]-Sigmatropic Rearrangement Reactions

Arnaud Voituriez, Lucie E. Zimmer and Andr

B. Charette

Publication Date (Web): January 22, 2010 (Article)

DOI: 10.1021/jo902618e

Cyclization Approaching to (−)-Lycojapodine A: Synthesis of Two Unnatural Alkaloids

Yu-Rong Yang, Liang Shen, Kun Wei and Qin-Shi Zhao

Publication Date (Web): January 22, 2010 (Note)

DOI: 10.1021/jo9026534

Synthesis of Medium-Bridged Twisted Lactams via Cation−π Control of the Regiochemistry of the Intramolecular Schmidt Reaction

Michal Szostak, Lei Yao and Jeffrey Aub

Publication Date (Web): January 22, 2010 (Article)

DOI: 10.1021/jo902574m

Intermediacy of Eudesmane Cation during Catalysis by Aristolochene Synthase

Juan A. Faraldos, Benson Kariuki and Rudolf K. Allemann

Publication Date (Web): January 22, 2010 (Article)

DOI: 10.1021/jo902397v

Synthesis of the Conformationally Constrained Tyrosine Analogues, (R)- and (S)-5-Hydroxy-2-aminoindan-2-carboxylic Acids

Francis N. Murigi, Gary S. Nichol and Eugene A. Mash

Publication Date (Web): January 22, 2010 (Note)

DOI: 10.1021/jo902438s

Self-Assembling Cyclic Tetrapeptide from Alternating C-Linked Carbo-β-amino Acid [(S)-β-Caa] and α-Aminoxy Acid [(R)-Ama]: A Selective Chloride Ion Receptor

Gangavaram V. M. Sharma, Vennampalli Manohar, Samit Kumar Dutta, Bojja Sridhar, Venna Ramesh, Ragampeta Srinivas and Ajit C. Kunwar

Publication Date (Web): January 22, 2010 (Article)

DOI: 10.1021/jo901923q

On the Origins of Diastereoselectivity in the Alkylation of Enolates Derived from N-1-(1′-Naphthyl)ethyl-O-tert-butylhydroxamates: Chiral Weinreb Amide Equivalents

Stephen G. Davies, Christopher J. Goodwin, David Hepworth, Paul M. Roberts and James E. Thomson

Publication Date (Web): January 22, 2010 (Article)

DOI: 10.1021/jo902499s

Rhodium(I)-Catalyzed Cycloisomerization of 1,6-Enynes to Bicyclo[4.1.0]heptenes

Sun Young Kim and Young Keun Chung

Publication Date (Web): January 22, 2010 (Note)

DOI: 10.1021/jo902273x

Mechanistic Pathways in CF₃COOH-Mediated Deacetalization Reactions

Wei Li, Jianchang Li, Yuchuan Wu, Nathan Fuller and Michelle A. Markus

Publication Date (Web): January 22, 2010 (Article)

DOI: 10.1021/jo902014z

Enantioselective Henry Reaction Catalyzed by Cu^II Salt and Bipiperidine

Artur Noole, Kristin Lippur, Andrus Metsala, Margus Lopp and T

nis Kanger

Publication Date (Web): January 22, 2010 (Note)

DOI: 10.1021/jo902664v

January 21, 2010

Gold- and Platinum-Catalyzed Formal Markownikoff’s Double Hydroamination of Alkynes: A Rapid Access to Tetrahydroquinazolinones and Angularly-Fused Analogues Thereof

Nitin T. Patil, Rahul D. Kavthe, Vivek S. Raut, Valmik S. Shinde and Balasubramanian Sridhar

Publication Date (Web): January 21, 2010 (Note)

DOI: 10.1021/jo902293f

January 20, 2010

Structure Elucidation of Dimethylformamide-Solvated Alkylzinc Cations in the Gas Phase

Frank Dreiocker, Jos Oomens, Anthony J. H. M. Meijer, Barry T. Pickup, Richard F. W. Jackson and Mathias Sch

fer

Publication Date (Web): January 20, 2010 (Article)

DOI: 10.1021/jo902492z

Unexpected Domino Reaction via Pd-Catalyzed Sonogashira Coupling of Benzimidoyl Chlorides with 1,6-Enynes and Cyclization To Synthesize Quinoline Derivatives

Guo-Lin Gao, Yan-Ning Niu, Ze-Yi Yan, Hong-Li Wang, Gang-Wei Wang, Ali Shaukat and Yong-Min Liang

Publication Date (Web): January 20, 2010 (Note)

DOI: 10.1021/jo9026116

Palladium-Catalyzed Preparation of Weinreb Amides from Boronic Acids and N-Methyl-N-methoxycarbamoyl Chloride

Ravi Krishnamoorthy, Sang Q. Lam, Christopher M. Manley and R. Jason Herr

Publication Date (Web): January 20, 2010 (Article)

DOI: 10.1021/jo902647h

Expanded Scope of Synthetic Bacteriochlorins via Improved Acid Catalysis Conditions and Diverse Dihydrodipyrrin-Acetals

Michael Krayer, Marcin Ptaszek, Han-Je Kim, Kelly R. Meneely, Dazhong Fan, Kristen Secor and Jonathan S. Lindsey

Publication Date (Web): January 20, 2010 (Featured Article)

DOI: 10.1021/jo9025572

Mild and Efficient Desymmetrization of Diynes via Hydroamination: Application to the Synthesis of (±)-Monomorine I

Vijaya Bhaskara Reddy Iska, Vincenzo Verdolino, Olaf Wiest and Paul Helquist

Publication Date (Web): January 20, 2010 (Note)

DOI: 10.1021/jo902674j

January 19, 2010

Highly Effective Vinylogous Mukaiyama−Michael Reaction Catalyzed by Silyl Methide Species Generated from 1,1,3,3-Tetrakis(trifluoromethanesulfonyl)propane

Arata Takahashi, Hikaru Yanai, Min Zhang, Takaaki Sonoda, Masaaki Mishima and Takeo Taguchi

Publication Date (Web): January 19, 2010 (Article)

DOI: 10.1021/jo902641g

Organocatalytic Enantioselective Synthesis of Both Diastereomers of α-Hydroxyphosphinates

Sampak Samanta, Sandun Perera and Cong-Gui Zhao

Publication Date (Web): January 19, 2010 (Article)

DOI: 10.1021/jo9022099

Brønsted Base-Catalyzed One-Pot Three-Component Biginelli-Type Reaction: An Efficient Synthesis of 4,5,6-Triaryl-3,4-dihydropyrimidin-2(1H)-one and Mechanistic Study

Zhi-Liang Shen, Xiao-Ping Xu and Shun-Jun Ji

Publication Date (Web): January 19, 2010 (Article)

DOI: 10.1021/jo902394y

January 14, 2010

Room Temperature Direct Alkynylation of 1,3,4-Oxadiazoles with Alkynyl Bromides under Copper Catalysis

Tsuyoshi Kawano, Naoto Matsuyama, Koji Hirano, Tetsuya Satoh and Masahiro Miura

Publication Date (Web): January 14, 2010 (Note)

DOI: 10.1021/jo9025622

Gold(III)-Catalyzed Tandem Reaction of Ketones with Phenols: Efficient and Highly Selective Synthesis of Functionalized 4H-Chromenes

Yunkui Liu, Jianqiang Qian, Shaojie Lou, Jie Zhu and Zhenyuan Xu

Publication Date (Web): January 14, 2010 (Note)

DOI: 10.1021/jo902619x

Modulating Reactivity and Diverting Selectivity in Palladium-Catalyzed Heteroaromatic Direct Arylation Through the Use of a Chloride Activating/Blocking Group

Beno

t Li

gault, Ivan Petrov, Serge I. Gorelsky and Keith Fagnou

Publication Date (Web): January 14, 2010 (Featured Article)

DOI: 10.1021/jo902515z

A Molecular Reel: Shuttling of a Rotor by Tumbling of a Macrocycle

Kazuhiro Yamauchi, Atsuhisa Miyawaki, Yoshinori Takashima, Hiroyasu Yamaguchi and Akira Harada

Publication Date (Web): January 14, 2010 (Featured Article)

DOI: 10.1021/jo902393n

On the Causes of Potential Inversion in 1,2,4,5-Tetrakis(amino)benzenes

Christopher J. Adams, Rosenildo C. da Costa, Ruth Edge, Dennis H. Evans and Matthew F. Hood

Publication Date (Web): January 14, 2010 (Article)

DOI: 10.1021/jo902411b

Total Syntheses of (−)-Fructigenine A and (−)-5-N-Acetylardeemin

Satoshi Takiguchi, Toshimasa Iizuka, Yuh-suke Kumakura, Kohta Murasaki, Naoko Ban, Kazuhiro Higuchi and Tomomi Kawasaki

Publication Date (Web): January 14, 2010 (Article)

DOI: 10.1021/jo9023107

Self-Assembly of C₃-Symmetrical Hexaaryltriindoles Driven by Solvophobic and CH−π Interactions

Eva M. Garc

a-Frutos, Gunther Hennrich, Enrique Gutierrez, Angeles Monge and Berta G

mez-Lor

Publication Date (Web): January 14, 2010 (Article)

DOI: 10.1021/jo902013v

January 12, 2010

OsO₄-Mediated Dihydroxylation of meso-Tetraphenylporphyrin N-Oxide and Transformation of the Resulting Diolchlorin N-Oxide Regioisomers

Subhadeep Banerjee, Matthias Zeller and Christian Br

ckner

Publication Date (Web): January 12, 2010 (Article)

DOI: 10.1021/jo9024286

January 11, 2010

Stereocontrolled Syntheses of (−)-Cubebol and (−)-10-Epicubebol Involving Intramolecular Cyclopropanation of α-Lithiated Epoxides

David M. Hodgson, Saifullah Salik and David J. Fox

Publication Date (Web): January 11, 2010 (Article)

DOI: 10.1021/jo9022974

December 29, 2009

Enzyme Catalysis by Hydrogen Bonds: The Balance between Transition State Binding and Substrate Binding in Oxyanion Holes

Luis Sim

n and Jonathan M. Goodman

Publication Date (Web): December 29, 2009 (Article)

DOI: 10.1021/jo901503d

December 18, 2009

Nanometer-Scale Water-Soluble Macrocycles from Nanometer-Sized Amino Acids

Chris M. Gothard and James S. Nowick

Publication Date (Web): December 18, 2009 (Article)

DOI: 10.1021/jo902268x

December 15, 2009

Metal-Catalyzed Cycloisomerization Reactions of cis-4-Hydroxy-5-alkynylpyrrolidinones and sis-5-Hydroxy-6-alkynylpiperidinones: Synthesis of Furo[3,2-b]pyrroles and Furo[3,2-b]pyridines

Jasmine C. Jury, Nalivela Kumara Swamy, Arife Yazici, Ian R. Morgan, Anthony C. Willis and Stephen G. Pyne

Publication Date (Web): December 15, 2009 (Addition/Correction)

DOI: 10.1021/jo9025385

December 14, 2009

Efficient Synthesis of 2-(Trimethylsilyl)phenyl Trifluoromethanesulfonate: A Versatile Precursor to o-Benzyne

Sarah M. Bronner and Neil K. Garg

Publication Date (Web): December 14, 2009 (Addition/Correction)

DOI: 10.1021/jo9025513

December 8, 2009

Theoretical and NMR Studies of Deuterium Isotopic Perturbation of Hydrogen Bonding in Symmetrical Dihydroxy Compounds

Daniel J. O'Leary, Daniel D. Hickstein, Bjarke K. V. Hansen and Poul Erik Hansen

Publication Date (Web): December 8, 2009 (Featured Article)

DOI: 10.1021/jo902075z

December 7, 2009

Glycosylation Using Unprotected Alkynyl Donors

Sreeman K. Mamidyala and M.G. Finn

Publication Date (Web): December 7, 2009 (Addition/Correction)

DOI: 10.1021/jo902465t

November 25, 2009

An Improved Synthesis of the Selective EP4 Receptor Agonist ONO-4819

Chisa Ohta, Shin-itsu Kuwabe, Tai Shiraishi, Ikuo Shinohara, Hiroshi Araki, Shigeru Sakuyama, Takayuki Makihara, Yasufumi Kawanaka, Shuichi Ohuchida and Takuya Seko

Publication Date (Web): November 25, 2009 (Addition/Correction)

DOI: 10.1021/jo902446x