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November 20, 2009

Synthesis of the Macrocyclic Core of Iriomoteolide 3a

Chada Raji Reddy, Gajula Dharmapuri and Nagavaram Narsimha Rao
Publication Date (Web): November 20, 2009 (Letter)

November 19, 2009

Copper-Catalyzed Tandem Nucleophilic Ring-Opening/Intramolecular Oxidative Amidation of N-Tosylaziridines and Hydrazones under Aerobic Conditions

Deng Hong, Xufeng Lin, Yuanxun Zhu, Ming Lei and Yanguang Wang
Publication Date (Web): November 19, 2009 (Letter)
DOI: 10.1021/ol902376w

Increased Yields and Simplified Purification with a Second-Generation Cobalt Catalyst for the Oxidative Formation of trans-THF Rings

Cory Palmer, Nicholas A. Morra, Andrew C. Stevens, Barbora Bajtos, Ben P. Machin and Brian L. Pagenkopf
Publication Date (Web): November 19, 2009 (Letter)
DOI: 10.1021/ol9023375

Palladium-Catalyzed Aryl C−H Bonds Activation/Acetoxylation Utilizing a Bidentate System

Fa-Rong Gou, Xiang-Chuan Wang, Peng-Fei Huo, Hai-Peng Bi, Zheng-Hui Guan and Yong-Min Liang
Publication Date (Web): November 19, 2009 (Letter)
DOI: 10.1021/ol902497k

Organozinc Generation via the Titanium-Catalyzed Activation of Alkyl Halides

Lauren M. Fleury and Brandon L. Ashfeld
Publication Date (Web): November 19, 2009 (Letter)
DOI: 10.1021/ol902374v

Highly Regioselective Palladium-Catalyzed Oxidative Coupling of Indolizines and Vinylarenes via C−H Bond Cleavage

Yuzhu Yang, Kai Cheng and Yuhong Zhang
Publication Date (Web): November 19, 2009 (Letter)
DOI: 10.1021/ol902315w

An Aldol Approach to the Total Synthesis of Pamamycin 621 A

Guo-Bao Ren and Yikang Wu
Publication Date (Web): November 19, 2009 (Letter)
DOI: 10.1021/ol902290v

November 18, 2009

Synthesis and Biological Activity of Oxa-Lacticin A2, a Lantibiotic Analogue with Sulfur Replaced by Oxygen

Hongqiang Liu, Vijaya R. Pattabiraman and John C. Vederas
Publication Date (Web): November 18, 2009 (Letter)
DOI: 10.1021/ol9025205

Silver-Catalyzed Protodecarboxylation of Heteroaromatic Carboxylic Acids

Pengfei Lu, Carolina Sanchez, Josep Cornella and Igor Larrosa
Publication Date (Web): November 18, 2009 (Letter)
DOI: 10.1021/ol902482p

Regiospecific Decarboxylative Allylation of Nitriles

Antonio Recio, III and Jon A. Tunge
Publication Date (Web): November 18, 2009 (Letter)
DOI: 10.1021/ol902065p

The Trichloromethide and Bromodichloromethide Carbanions

Robert A. Moss, Min Zhang and Karsten Krogh-Jespersen
Publication Date (Web): November 18, 2009 (Letter)
DOI: 10.1021/ol902479x

Microwave-Assisted Domino and Multicomponent Reactions with Cyclic Acylketenes: Expeditious Syntheses of Oxazinones and Oxazindiones

Marc Presset, Yoann Coquerel and Jean Rodriguez
Publication Date (Web): November 18, 2009 (Letter)
DOI: 10.1021/ol9024056

Regioselective Iron-Catalyzed Decarboxylative Allylic Etherification

Rushi Trivedi and Jon A. Tunge
Publication Date (Web): November 18, 2009 (Letter)
DOI: 10.1021/ol902291z

Brucine-Derived Amino Alcohol Catalyzed Asymmetric Henry Reaction: An Orthogonal Enantioselectivity Approach

Hun Young Kim and Kyungsoo Oh
Publication Date (Web): November 18, 2009 (Letter)
DOI: 10.1021/ol902380z

Reaction-Based Fluorescent Sensing of Au(I)/Au(III) Species: Mechanistic Implications on Vinylgold Intermediates

Olga A. Egorova, Hyewon Seo, Amrita Chatterjee and Kyo Han Ahn
Publication Date (Web): November 18, 2009 (Letter)
DOI: 10.1021/ol902395x

Phorbaketals A, B, and C, Sesterterpenoids with a Spiroketal of Hydrobenzopyran Moiety Isolated from the Marine Sponge Phorbas sp.

Jung-Rae Rho, Buyng Su Hwang, Chung Ja Sim, Seewon Joung, Hee-Yoon Lee and Hyeon-Jin Kim
Publication Date (Web): November 18, 2009 (Letter)
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Chiral 1,2-Diols: The Assignment of Their Absolute Configuration by NMR Made Easy

Flix Freire, Jos Manuel Seco, Emilio Quio and Ricardo Riguera
Publication Date (Web): November 18, 2009 (Letter)
DOI: 10.1021/ol9021639

A New Organocatalyzed Michael−Michael Cascade Reaction Generates Highly Substituted Fused Carbocycles

Patrick G. McGarraugh and Stacey E. Brenner
Publication Date (Web): November 18, 2009 (Letter)
DOI: 10.1021/ol9024293

A Gold(III) Ion-Selective Fluorescent Probe and Its Application to Bioimagings

Young-Keun Yang, Sunho Lee and Jinsung Tae
Publication Date (Web): November 18, 2009 (Letter)
DOI: 10.1021/ol902325u

Alasmontamine A, A First Tetrakis Monoterpene Indole Alkaloid from Tabernaemontana elegans

Yusuke Hirasawa, Saori Miyama, Takahiro Hosoya, Koichiro Koyama, Abdul Rahman, Idha Kusumawati, Noor Cholies Zaini and Hiroshi Morita
Publication Date (Web): November 18, 2009 (Letter)

Unexpected Multiple Electrophilic Addition Reaction of (Z)-Alk-2-en-4-ynoates with N,N-Dibromo-p-toluenesulfonamide (TsNBr2): A Highly Diastereoselective Synthesis of Densely Functionalized Aziridines

Ruwei Shen and Xian Huang
Publication Date (Web): November 18, 2009 (Letter)
DOI: 10.1021/ol902446h

November 17, 2009

Cooperativity of Regiochemistry Control Strategies in Reductive Couplings of Propargyl Alcohols and Aldehydes

Hasnain A. Malik, Mani Raj Chaulagain and John Montgomery
Publication Date (Web): November 17, 2009 (Letter)
DOI: 10.1021/ol902561r

First Total Synthesis of Tubulysin B

Orlando Pando, Simon Drner, Rainer Preusentanz, Annika Denkert, Andrea Porzel, Wolfgang Richter and Ludger Wessjohann
Publication Date (Web): November 17, 2009 (Letter)

Molecular Machinery: Synthesis of a “Nanodragster”

Guillaume Vives, JungHo Kang, Kevin F. Kelly and James M. Tour
Publication Date (Web): November 17, 2009 (Letter)
DOI: 10.1021/ol902312m

A Concise Route to the Proposed Structure of Lydiamycin B, an Antimycobacterial Depsipeptide

Wenhua Li, Jiangang Gan and Dawei Ma
Publication Date (Web): November 17, 2009 (Letter)
DOI: 10.1021/ol9024474

Oxygen- and Sulfur-Containing Positively Charged Polycyclic Aromatic Hydrocarbons

Dongqing Wu, Wojciech Pisula, Monika C. Haberecht, Xinliang Feng and Klaus Mllen
Publication Date (Web): November 17, 2009 (Letter)
DOI: 10.1021/ol902366y

Total Synthesis of Polyrhacitides A and B by Use of an Iterative Strategy for the Stereoselective Synthesis of 1,3-Polyol Arrays

Helge Menz and Stefan F. Kirsch
Publication Date (Web): November 17, 2009 (Letter)
DOI: 10.1021/ol902135v

EPR and NMR Investigation on the Interactions of Nitroxide Probes with Resorcin[4]arene Molecular Capsules

Song Yi, Elisabetta Mileo and Angel E. Kaifer
Publication Date (Web): November 17, 2009 (Letter)
DOI: 10.1021/ol902391u

November 16, 2009

Suppressed β-Effect of Silicon in 3-Silylated Monocyclic β-Lactams: The Role of Antiaromaticity

Subhendu Sekhar Bag, Rajen Kundu, Amit Basak and Zdenek Slanina
Publication Date (Web): November 16, 2009 (Letter)

November 13, 2009

Novel Nucleophilic Heterocyclic Carbene Mediated Stereoselective Conjugate Addition of Enals to Nitrostyrenes via Homoenolate

Vijay Nair, C. R. Sinu, Beneesh P. Babu, Vimal Varghese, Anu Jose and Eringathodi Suresh
Publication Date (Web): November 13, 2009 (Letter)
DOI: 10.1021/ol901918x

Anhydrous Hydration of Nitriles to Amides using Aldoximes as the Water Source

Jinwoo Lee, Min Kim, Sukbok Chang and Hee-Yoon Lee
Publication Date (Web): November 13, 2009 (Letter)
DOI: 10.1021/ol902309z

Highly Enantioselective Ketone-Ene Reactions of Trifluoropyruvate: Significant Counterion Effect of the In(III)−PyBox Complex

Jun-Feng Zhao, Teguh-Budiono W. Tjan, Boon-Hong Tan and Teck-Peng Loh
Publication Date (Web): November 13, 2009 (Letter)
DOI: 10.1021/ol902507x

Dramatic Effect of Solvent Hydrogen Bond Basicity on the Regiochemistry of SNAr Reactions of Electron-Deficient Polyfluoroarenes

Xiaolun Wang, Edward J. Salaski, Dan M. Berger and Dennis Powell
Publication Date (Web): November 13, 2009 (Letter)
DOI: 10.1021/ol902353t

Microwave-Assisted Synthesis of 2′-O-Aryluridine Derivatives

Yusuke Oeda, Yoshihiro Iijima, Haruhiko Taguchi, Akihiro Ohkubo, Khoji Seio and Mitsuo Sekine
Publication Date (Web): November 13, 2009 (Letter)
DOI: 10.1021/ol902142w
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November 12, 2009

Highly Catalytic Asymmetric Addition of Deactivated Alkyl Grignard Reagents to Aldehydes

Chao-Shan Da, Jun-Rui Wang, Xiao-Gang Yin, Xin-Yuan Fan, Yi Liu and Sheng-Li Yu
Publication Date (Web): November 12, 2009 (Letter)

Ambient Temperature Hydrophosphination of Internal, Unactivated Alkynes and Allenyl Phosphineoxides with Phosphine Borane Complexes

Carl A. Busacca, Elisa Farber, Jay DeYoung, Scot Campbell, Nina C. Gonnella, Nelu Grinberg, Nizar Haddad, Heewon Lee, Shengli Ma, Diana Reeves, Sherry Shen and Chris H. Senanayake
Publication Date (Web): November 12, 2009 (Letter)

General and Functional Group-Tolerable Approach to Allenylsilanes by Rhodium-Catalyzed Coupling between Propargylic Carbonates and a Silylboronate

Hirohisa Ohmiya, Hideto Ito and Masaya Sawamura
Publication Date (Web): November 12, 2009 (Letter)

Carbonyldiimidazole-Mediated Lossen Rearrangement

Pascal Dub, Noah F. Fine Nathel, Michael Vetelino, Michel Couturier, Claude Larrive Aboussafy, Simon Pichette, Matthew L. Jorgensen and Mark Hardink
Publication Date (Web): November 12, 2009 (Letter)
DOI: 10.1021/ol9023387

Synthesis of Carbamates from Diethoxycarbonyl Hydrazine Derivatives by E1cB Eliminative Cleavage of the N−N′-Bond Rather than Reduction

Philip Magnus, Negar Garizi, Kimberly A. Seibert and Alexandra Ornholt
Publication Date (Web): November 12, 2009 (Letter)

Palladium-Catalyzed Decarboxylative [4 + 3] Cyclization of γ-Methylidene-δ-valerolactones with 1,1-Dicyanocyclopropanes

Ryo Shintani, Masataka Murakami, Takaoki Tsuji, Hideyuki Tanno and Tamio Hayashi
Publication Date (Web): November 12, 2009 (Letter)
DOI: 10.1021/ol902326s

November 11, 2009

Pd(II)/tBu-quinolineoxazoline: An Air-Stable and Modular Chiral Catalyst System for Enantioselective Oxidative Cascade Cyclization

Wei He, Kai-Tai Yip, Nian-Yong Zhu and Dan Yang
Publication Date (Web): November 11, 2009 (Letter)
DOI: 10.1021/ol902348t

Facile Synthesis of Substituted 5-Amino- and 3-Amino-1,2,4-Thiadiazoles from a Common Precursor

Paul M. Wehn, Paul E. Harrington and John E. Eksterowicz
Publication Date (Web): November 11, 2009 (Letter)
DOI: 10.1021/ol902371y

Bromo-Directed N-2 Alkylation of NH-1,2,3-Triazoles: Efficient Synthesis of Poly-Substituted 1,2,3-Triazoles

Xiao-jun Wang, Kanwar Sidhu, Li Zhang, Scot Campbell, Nizar Haddad, Diana C. Reeves, Dhileepkumar Krishnamurthy and Chris H. Senanayake
Publication Date (Web): November 11, 2009 (Letter)
DOI: 10.1021/ol902334x

Modular Construction of 2-Substituted Benzo[b]furans from 1,2-Dichlorovinyl Ethers

Laina M. Geary and Philip G. Hultin
Publication Date (Web): November 11, 2009 (Letter)
DOI: 10.1021/ol902307m

Daphhimalenine A, a New Alkaloid with an Unprecedented Skeleton, from Daphniphyllum himalense

Yu Zhang, Ying-Tong Di, Qiang Zhang, Shu-Zhen Mu, Cheng-Jian Tan, Xin Fang, Hong-Ping He, Shun-Lin Li and Xiao-Jiang Hao
Publication Date (Web): November 11, 2009 (Letter)
DOI: 10.1021/ol902262g

Asymmetric Construction of Rings A−D of Daphnicyclidin-Type Alkaloids

Travis B. Dunn, J. Michael Ellis, Christiane C. Kofink, James R. Manning and Larry E. Overman
Publication Date (Web): November 11, 2009 (Letter)
DOI: 10.1021/ol902373m

4-Fluoro-2,4-methanoproline

Anton N. Tkachenko, Dmytro S. Radchenko, Pavel K. Mykhailiuk, Oleksandr O. Grygorenko and Igor V. Komarov
Publication Date (Web): November 11, 2009 (Letter)
DOI: 10.1021/ol902381w

Boron-Catalyzed Direct Aldol Reactions of Pyruvic Acids

Doris Lee, Stephen G. Newman and Mark S. Taylor
Publication Date (Web): November 11, 2009 (Letter)
DOI: 10.1021/ol902322r

Selective Synthesis of Eight-Membered Cyclic Ureas by the [6 + 2] Cycloaddition Reaction of 2-Vinylazetidines and Electron-Deficient Isocyanates

Shunsuke Koya, Kenichi Yamanoi, Ryu Yamasaki, Isao Azumaya, Hyuma Masu and Shinichi Saito
Publication Date (Web): November 11, 2009 (Letter)
DOI: 10.1021/ol902299p

Benzo[cd]azulene Skeleton: Azulene, Heptafulvene, and Tropone Derivatives

Ingo B. Aumller and Jari Yli-Kauhaluoma
Publication Date (Web): November 11, 2009 (Letter)
DOI: 10.1021/ol902283q

Synthesis of (S)-Jamaicamide C Carboxylic Acid

Kristin M. Graf, Martin G. Tabor, Milton L. Brown and Mikell Paige
Publication Date (Web): November 11, 2009 (Letter)
DOI: 10.1021/ol9021222

November 10, 2009

Convergent Synthesis of Fostriecin via Selective Alkene Couplings and Regioselective Asymmetric Dihydroxylation

Omar Robles and Frank E. McDonald
Publication Date (Web): November 10, 2009 (Letter)
DOI: 10.1021/ol902365n

Synthesis of Biphenyl Proteomimetics as Estrogen Receptor-α Coactivator Binding Inhibitors

Anna B. Williams, Patrick T. Weiser, Robert N. Hanson, Jillian R. Gunther and John A. Katzenellenbogen
Publication Date (Web): November 10, 2009 (Letter)
DOI: 10.1021/ol901999f

Concise Synthesis of Pauciflorol F Using a Larock Annulation

Jenna L. Jeffrey and Richmond Sarpong
Publication Date (Web): November 10, 2009 (Letter)
DOI: 10.1021/ol902141z

November 9, 2009

Total Synthesis and Structural Revision of the Presumed Aeruginosins 205A and B

Stephen Hanessian, Xiaotian Wang, Karolina Ersmark, Juan R. DelValle and Ellen Klegraf
Publication Date (Web): November 9, 2009 (Addition/Correction)
DOI: 10.1021/ol9025342

Origin of Thermodynamic versus Kinetic Control of Allene Hydroboration with 9-Borabicyclo[3.3.1]nonane and 10(R)-Trimethylsilyl-9-Borabicyclo[3.3.2]decane

Daniel H. Ess, Jeremy Kister, Ming Chen and William R. Roush
Publication Date (Web): November 9, 2009 (Letter)
DOI: 10.1021/ol902364d

Preparation of Zwitterionic Hydroquinone-Fused [1,4]Oxazinium Derivatives via a Photoinduced Intramolecular Dehydrogenative-Coupling Reaction

Chenyi Yi, Shi-Xia Liu, Antonia Neels, Philippe Renaud and Silvio Decurtins
Publication Date (Web): November 9, 2009 (Letter)
DOI: 10.1021/ol902355b

Catalytic Allylic C−H Acetoxylation and Benzoyloxylation via Suggested (η3-Allyl)palladium(IV) Intermediates

Lukasz T. Pilarski, Nicklas Selander, Dietrich Bse and Klmn J. Szab
Publication Date (Web): November 9, 2009 (Letter)
DOI: 10.1021/ol9023369

Enhancement of Reaction Efficiency by Functionalized Alcohols on Gold(I)-Catalyzed Intermolecular Hydroalkoxylation of Unactivated Olefins

Toshifumi Hirai, Akiyuki Hamasaki, Aki Nakamura and Makoto Tokunaga
Publication Date (Web): November 9, 2009 (Letter)
DOI: 10.1021/ol9023166

Two Novel Carbazole Dyes for Dye-Sensitized Solar Cells with Open-Circuit Voltages up to 1 V Based on Br−/Br3− Electrolytes

Chao Teng, Xichuan Yang, Chunze Yuan, Chaoyan Li, Ruikui Chen, Haining Tian, Shifeng Li, Anders Hagfeldt and Licheng Sun
Publication Date (Web): November 9, 2009 (Letter)
DOI: 10.1021/ol9022936

Competitive Formation of N-Diazeniumdiolates and N-Nitrosamines via Anaerobic Reactions of Polyamines with Nitric Oxide

Peter N. Coneski and Mark H. Schoenfisch
Publication Date (Web): November 9, 2009 (Letter)
DOI: 10.1021/ol902282y

Desymmetrization of Cyclic meso-Epoxides with Silicon Tetrachloride Catalyzed by PINDOX, a Chiral Bipyridine Mono-N-oxide

Andrei V. Malkov, Malcolm R. Gordon, Sigitas Stonius, Javid Hussain and Pavel Koovsk
Publication Date (Web): November 9, 2009 (Letter)
DOI: 10.1021/ol902148s

Acryloyl Chloride: An Excellent Substrate for Cross-Metathesis. A One-Pot Sequence for the Synthesis of Substituted α,β-Unsaturated Carbonyl Derivatives

Laurent Ferri, Samir Bouzbouz and Janine Cossy
Publication Date (Web): November 9, 2009 (Letter)
DOI: 10.1021/ol9021386

November 6, 2009

Jatrophalactam, A Novel Diterpenoid Lactam Isolated from Jatropha curcas

Xia-Chang Wang, Zong-Ping Zheng, Xian-Wen Gan and Li-Hong Hu
Publication Date (Web): November 6, 2009 (Letter)
DOI: 10.1021/ol902349f

Asymmetric Total Syntheses of (−)-Renieramycin M and G and (−)-Jorumycin Using Aziridine as a Lynchpin

Yan-Chao Wu and Jieping Zhu
Publication Date (Web): November 6, 2009 (Letter)
DOI: 10.1021/ol9024919

November 5, 2009

A Novel Heterocyclic Scaffold Formed by Ring Expansion of a Cyclic Sulfone to Sulfonamides

Magnus Sellstedt and Fredrik Almqvist
Publication Date (Web): November 5, 2009 (Letter)
DOI: 10.1021/ol9023024

First Asymmetric Total Syntheses of Fawcettimine-Type Lycopodium Alkaloids, Lycoposerramine-C and Phlegmariurine-A

Atsushi Nakayama, Noriyuki Kogure, Mariko Kitajima and Hiromitsu Takayama
Publication Date (Web): November 5, 2009 (Letter)
DOI: 10.1021/ol902437t

Regioselective Nucleophilic Addition to Pyridinium Salts: A New Route to Substituted Dihydropyridones

Timothy J. Donohoe, Matthew J. Connolly and Lesley Walton
Publication Date (Web): November 5, 2009 (Letter)

Stereoselective Synthesis of Donor−Acceptor Substituted Cyclopropafuranones by Intramolecular Cyclopropanation of Vinylogous Carbonates: Divergent Synthesis of Tetrahydrofuran-3-one, Tetrahydropyran-3-one, and Lactones

Santosh J. Gharpure, Manoj K. Shukla and U. Vijayasree
Publication Date (Web): November 5, 2009 (Letter)
DOI: 10.1021/ol902301h

November 4, 2009

Stereocontrolled Access to Unsymmetrical 1,1-Diaryl-2-fluoroethenes

Grgory Landelle, Marc-Olivier Turcotte-Savard, Judikalle Marterer, Pier Alexandre Champagne and Jean-Franois Paquin
Publication Date (Web): November 4, 2009 (Letter)
DOI: 10.1021/ol9022672

Stereoselective Synthesis of (E)-2-En-4-ynoic Acids with Ynolates: Catalytic Conversion to Tetronic Acids and 2-Pyrones

Takashi Yoshikawa and Mitsuru Shindo
Publication Date (Web): November 4, 2009 (Letter)
DOI: 10.1021/ol902086t

Highly Efficient Cyanoimidation of Aldehydes

Ping Yin, Wen-Bo Ma, Yue Chen, Wen-Cai Huang, Yong Deng and Ling He
Publication Date (Web): November 4, 2009 (Letter)
DOI: 10.1021/ol902207h

Oxidative Carbon−Carbon Bond Formation via Allyldimethylsilyl Enol Ethers

Leah C. Konkol, Brian T. Jones and Regan J. Thomson
Publication Date (Web): November 4, 2009 (Letter)

Apoptolidins E and F, New Glycosylated Macrolactones Isolated from Nocardiopsis sp.

Paul A. Wender and Kate E. Longcore
Publication Date (Web): November 4, 2009 (Letter)
DOI: 10.1021/ol902308v

A Core-Substituted Naphthalene Diimide Fluoride Sensor

Sheshanath V. Bhosale, Sidhanath V. Bhosale, Mohan B. Kalyankar and Steven J. Langford
Publication Date (Web): November 4, 2009 (Letter)
DOI: 10.1021/ol9022722

November 3, 2009

Aryl Hydrazide beyond as Surrogate of Aryl Hydrazine in the Fischer Indolization: The Synthesis of N-Cbz-indoles, N-Cbz-carbazoles, and N,N′-Bis-Cbz-pyrrolo[2,3-f]indoles

In-Keol Park, Sung-Eun Suh, Byeong-Yun Lim and Cheon-Gyu Cho
Publication Date (Web): November 3, 2009 (Letter)
DOI: 10.1021/ol902250x

Chiral Brønsted Acid-Catalyzed Enantioselective Multicomponent Mannich Reaction: Synthesis of anti-1,3-Diamines Using Enecarbamates as Nucleophiles

Guillaume Dagousset, Fleur Drouet, Graldine Masson and Jieping Zhu
Publication Date (Web): November 3, 2009 (Letter)
DOI: 10.1021/ol9023985

November 2, 2009

A New Ring Closure Approach to Enantiopure 3,6-Dihydro-2H-pyrans: Stereodivergent Access to Carbohydrate Mimetics

Fabian Pfrengle, Dieter Lentz and Hans-Ulrich Reissig
Publication Date (Web): November 2, 2009 (Letter)
DOI: 10.1021/ol902354f

Direct Meta-Selective Alkylation of Perylene Bisimides via Palladium-Catalyzed C−H Functionalization

Wan Yue, Yan Li, Wei Jiang, Yonggang Zhen and Zhaohui Wang
Publication Date (Web): November 2, 2009 (Letter)
DOI: 10.1021/ol9023198

Palladium-Catalyzed Cross-Coupling Reaction of Secondary Benzylic Bromides with Grignard Reagents

Ana Lpez-Prez, Javier Adrio and Juan C. Carretero
Publication Date (Web): November 2, 2009 (Letter)
DOI: 10.1021/ol902335c

New Building Block for C3 Symmetry Molecules: Synthesis of s-Triazine-Based Redox Active Chromophores

Anglica Garca, Braulio Insuasty, Mangeles Herranz, Roberto Martnez-lvarez and Nazario Martn
Publication Date (Web): November 2, 2009 (Letter)
DOI: 10.1021/ol902203t

Synthesis of Arylated Perylene Bisimides through C−H Bond Cleavage under Ruthenium Catalysis

Satomi Nakazono, Shanmugam Easwaramoorthi, Dongho Kim, Hiroshi Shinokubo and Atsuhiro Osuka
Publication Date (Web): November 2, 2009 (Letter)
DOI: 10.1021/ol902271b

Lodopyridone, a Structurally Unprecedented Alkaloid from a Marine Actinomycete

Katherine N. Maloney, John B. MacMillan, Christopher A. Kauffman, Paul R. Jensen, Antonio G. DiPasquale, Arnold L. Rheingold and William Fenical
Publication Date (Web): November 2, 2009 (Letter)
DOI: 10.1021/ol901997k

Synthesis of All Diastereomers of the Piperidine−Alkaloid Substructure of Cyclopamine

Philipp Heretsch, Sebastian Rabe and Athanassios Giannis
Publication Date (Web): November 2, 2009 (Letter)
DOI: 10.1021/ol902270f

Azide Conjugatable and pH Responsive Near-Infrared Fluorescent Imaging Probes

Julie Murtagh, Daniel O. Frimannsson and Donal F. O’Shea
Publication Date (Web): November 2, 2009 (Letter)
DOI: 10.1021/ol902140v

October 30, 2009

Asymmetric Conjugate Reductions of Coumarins. A New Route to Tolterodine and Related Coumarin Derivatives

Brian D. Gallagher, Benjamin R. Taft and Bruce H. Lipshutz
Publication Date (Web): October 30, 2009 (Letter)
DOI: 10.1021/ol9020404

Substituted 1,4-Benzoxazepines, 1,5-Benzoxazocines, and N- and S-Variants

Janjira Rujirawanich and Timothy Gallagher
Publication Date (Web): October 30, 2009 (Letter)
DOI: 10.1021/ol9023453

Intermolecular Decarboxylative Direct C-3 Arylation of Indoles with Benzoic Acids

Josep Cornella, Pengfei Lu and Igor Larrosa
Publication Date (Web): October 30, 2009 (Letter)
DOI: 10.1021/ol902304n

Smiles Rearrangement as a Tool for the Preparation of Dihydrodipyridopyrazines

Oana-Irina Patriciu, Adriana-Luminita Fînaru, Stphane Massip, Jean-Michel Leger, Christian Jarry and Grald Guillaumet
Publication Date (Web): October 30, 2009 (Letter)
DOI: 10.1021/ol902369v

Stereoselective Synthesis of (E)-(Trisubstituted alkenyl)borinic Esters: Stereochemistry Reversed by Ligand in the Palladium-Catalyzed Reaction of Alkynylborates with Aryl Halides

Naoki Ishida, Yasuhiro Shimamoto and Masahiro Murakami
Publication Date (Web): October 30, 2009 (Letter)
DOI: 10.1021/ol902278q

Regioselective Allene Synthesis and Propargylations with Propargyl Diethanolamine Boronates

Daniel R. Fandrick, Jonathan T. Reeves, Zhulin Tan, Heewon Lee, Jinhua J. Song, Nathan K. Yee and Chris H. Senanayake
Publication Date (Web): October 30, 2009 (Letter)
DOI: 10.1021/ol9022529

Nitrile Ylides: Diastereoselective Cycloadditions using Chiral Oxzolidinones Without Lewis Acid

Mukund P. Sibi, Takahiro Soeta and Craig P. Jasperse
Publication Date (Web): October 30, 2009 (Letter)
DOI: 10.1021/ol9018584

A Hypervalent Iodine-Induced Double Annulation Enables a Concise Synthesis of the Pentacyclic Core Structure of the Cortistatins

Jessica L. Frie, Christopher S. Jeffrey and Erik J. Sorensen
Publication Date (Web): October 30, 2009 (Letter)
DOI: 10.1021/ol902168g

Expedient Construction of the Ziegler Intermediate Useful for the Synthesis of Forskolin via Consecutive Rearrangements

Heping Ye, Gang Deng, Jun Liu and Fayang G. Qiu
Publication Date (Web): October 30, 2009 (Letter)
DOI: 10.1021/ol902133q

Convergent Synthesis of Stereodefined exo-Alkylidene-γ-Lactams from β-Halo Allylic Alcohols

Shuhei Umemura, Martin McLaughlin and Glenn C. Micalizio
Publication Date (Web): October 30, 2009 (Letter)
DOI: 10.1021/ol9022134

October 29, 2009

Total Synthesis of (±)-Cordypyridones A and B and Related Epimers

Ian L. Jones, Felicity K. Moore and Christina L. L. Chai
Publication Date (Web): October 29, 2009 (Letter)
DOI: 10.1021/ol9023437
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