Table of Contents

Journal Cover
September 6, 2001
Volume 3, Issue 18
Pages 2789-2939
For Selected Content:

Letters

Reductive Activation of Mitomycin A by Thiols

Manuel M. Paz and Maria Tomasz
pp 2789–2792
Publication Date (Web): August 15, 2001 (Letter)
DOI: 10.1021/ol015517+

The 5,6- and 4,5-Benzo Derivatives of 1-Hydroxy-7-azabenzotriazole

Louis A. Carpino and Fernando J. Ferrer
pp 2793–2795
Publication Date (Web): August 08, 2001 (Letter)
DOI: 10.1021/ol016063j

Solid-Phase Synthesis of 1,7-Disubstituted-1,3,5-triazepane-2,4-diones

Yongping Yu, John M. Ostresh, and Richard A. Houghten
pp 2797–2799
Publication Date (Web): August 11, 2001 (Letter)
DOI: 10.1021/ol010102+

The pH-Dependent Role of Superoxide in Riboflavin-Catalyzed Photooxidation of 8-Oxo-7,8-dihydroguanosine

Wenchen Luo, James G. Muller, and Cynthia J. Burrows
pp 2801–2804
Publication Date (Web): August 11, 2001 (Letter)
DOI: 10.1021/ol0161763

A Novel One-Pot Conversion of Aldehydes to Trifluoromethylated Bromoallylic Alcohols

Yanchang Shen and Yuming Zhang
pp 2805–2806
Publication Date (Web): August 14, 2001 (Letter)
DOI: 10.1021/ol010115n

Regiospecific Synthesis of 4-(2-Oxoalkyl)pyridines

Alan R. Katritzky, Suoming Zhang, Thomas Kurz, and Mingyi WangPeter J. Steel
pp 2807–2809
Publication Date (Web): August 16, 2001 (Letter)
DOI: 10.1021/ol010116f

Studies on the Total Synthesis of Tallysomycin. Synthesis of the Threonylbithiazole Moiety Containing a Structurally Unique Glycosylcarbinolamide

Marcos L. Sznaidman and Sidney M. Hecht
pp 2811–2814
Publication Date (Web): August 10, 2001 (Letter)
DOI: 10.1021/ol0101178

Structure, Histone Deacetylase, and Antiprotozoal Activities of Apicidins B and C, Congeners of Apicidin with Proline and Valine Substitutions

Sheo B. Singh, Deborah L. Zink, Jerrold M. Liesch, Anne W. Dombrowski, Sandra J. Darkin-Rattray, Dennis M. Schmatz, and Michael A. Goetz
pp 2815–2818
Publication Date (Web): August 15, 2001 (Letter)
DOI: 10.1021/ol016240g

Intramolecular [2 + 2]- Photocycloaddition/Thermal Fragmentation Approach toward 5−8−5 Ring Systems

Priscilla C.-K. Lo and Marc L. Snapper
pp 2819–2821
Publication Date (Web): August 10, 2001 (Letter)
DOI: 10.1021/ol016244l

Synthesis of N-(3-Arylpropyl)amino Acid Derivatives by Sonogashira Types of Reaction in Aqueous Media

M. Pilar López-Deber, Luis Castedo, and Juan R. Granja
pp 2823–2826
Publication Date (Web): August 10, 2001 (Letter)
DOI: 10.1021/ol0162421

A Streamlined Synthesis for 2,3-Dihydroxyterephthalamides

Christine J. Gramer and Kenneth N. Raymond
pp 2827–2830
Publication Date (Web): August 10, 2001 (Letter)
DOI: 10.1021/ol016253u

Regioselective Aromatic Borylation in an Inert Solvent

Man Kin Tse, Jian-Yang Cho, and Milton R. Smith, III
pp 2831–2833
Publication Date (Web): August 08, 2001 (Letter)
DOI: 10.1021/ol0162668

Mild Oxidative One-Pot Allyl Group Cleavage

Pavel I. Kitov and David R. Bundle
pp 2835–2838
Publication Date (Web): August 11, 2001 (Letter)
DOI: 10.1021/ol016278t

Generation of (E)-Silylketene Acetals in a Rhodium-DuPhos Catalyzed Two-Step Reductive Aldol Reaction

Cun-Xiang Zhao, Jonathan Bass, and James P. Morken
pp 2839–2842
Publication Date (Web): August 14, 2001 (Letter)
DOI: 10.1021/ol016279l

Synthesis of (+)-Galiellalactone. Absolute Configuration of Galiellalactone

Martin Johansson and Olov Sterner
pp 2843–2845
Publication Date (Web): August 04, 2001 (Letter)
DOI: 10.1021/ol016286+

Asymmetric Synthesis of Trifluoromethylated Allylic Amines Using α,β-Unsaturated N-tert-Butanesulfinimines

G. K. Surya Prakash, Mihirbaran Mandal, and George A. Olah
pp 2847–2850
Publication Date (Web): August 09, 2001 (Letter)
DOI: 10.1021/ol010134x

Ru-Catalyzed Cyclocarbonylation of α- and β-Allenic Sulfonamides:  Synthesis of γ- and δ-Unsaturated Lactams

Suk-Ku Kang, Kwang-Jin Kim, Chan-Mo Yu, Jeong-Wook Hwang, and Young-Kyu Do
pp 2851–2853
Publication Date (Web): August 07, 2001 (Letter)
DOI: 10.1021/ol016281c

Synthesis of Novel Derivatives of 1,4,7-Triazacyclononane

Andrew Warden, Bim Graham, Milton T. W. Hearn, and Leone Spiccia
pp 2855–2858
Publication Date (Web): August 15, 2001 (Letter)
DOI: 10.1021/ol016291d

Generating Diversity in Difluoromethyl Ketone Derivatives

Gareth A. DeBoos, Jeremy J. Fullbrook, and Jonathan M. Percy
pp 2859–2861
Publication Date (Web): August 09, 2001 (Letter)
DOI: 10.1021/ol010135p

Stereocontrolled Synthesis of the Northern Part of Potent Proteasome Inhibitor TMC-95A

Masayuki Inoue, Hidetomo Furuyama, Hayato Sakazaki, and Masahiro Hirama
pp 2863–2865
Publication Date (Web): August 11, 2001 (Letter)
DOI: 10.1021/ol016303v

Analogues of Bleomycin:  Synthesis of Conformationally Rigid Methylvalerates

Michael J. Rishel and Sidney M. Hecht
pp 2867–2869
Publication Date (Web): August 10, 2001 (Letter)
DOI: 10.1021/ol010139u

Copper-Mediated Cross-Coupling of Functionalized Arylmagnesium Reagents with Functionalized Alkyl and Benzylic Halides

Wolfgang Dohle, David M. Lindsay, and Paul Knochel
pp 2871–2873
Publication Date (Web): August 04, 2001 (Letter)
DOI: 10.1021/ol0163272

A Novel Three-Component Butenolide Synthesis

Barbara Beck, Marina Magnin-Lachaux, Eberhardt Herdtweck, and Alexander Dömling
pp 2875–2878
Publication Date (Web): August 04, 2001 (Letter)
DOI: 10.1021/ol016328u

Enantioselective Synthesis of a Mitosane Core Assisted by Diversity-Based Catalyst Discovery

Nikolaos Papaioannou, Catherine A. Evans, Jarred T. Blank, and Scott J. Miller
pp 2879–2882
Publication Date (Web): August 03, 2001 (Letter)
DOI: 10.1021/ol016372+

Synthesis of Diynes and Tetraynes from in Situ Desilylation/Dimerization of Acetylenes

Matthew A. Heuft, Shawn K. Collins, Glenn P. A. Yap, and Alex G. Fallis
pp 2883–2886
Publication Date (Web): August 15, 2001 (Letter)
DOI: 10.1021/ol016414u

Multiple-Electron Transfer in a Single Step. Design and Synthesis of Highly Charged Cation-Radical Salts

Rajendra Rathore, Carrie L. Burns, and Mihaela I. Deselnicu
pp 2887–2890
Publication Date (Web): August 09, 2001 (Letter)
DOI: 10.1021/ol0163474

[4 + 3] Cycloaddition of Cyclopropanone Hemiacetals1

Sung Yun Cho, Hyoung Ik Lee, and Jin Kun Cha
pp 2891–2893
Publication Date (Web): August 09, 2001 (Letter)
DOI: 10.1021/ol016354s

Facile Three-Component Coupling Procedure for the Synthesis of Substituted Tetrahydroisoindole-1,3-diones from α,β-Unsaturated Aldehydes

Axel Jacobi von Wangelin, Helfried Neumann, Dirk Gördes, Anke Spannenberg, and Matthias Beller
pp 2895–2898
Publication Date (Web): August 15, 2001 (Letter)
DOI: 10.1021/ol0101436

Concise Synthesis of a Lactonamycin Model System by Diastereoselective Dihydroxylation of a Highly Functionalized Naphthoquinone

Christopher Cox and Samuel J. Danishefsky
pp 2899–2902
Publication Date (Web): August 07, 2001 (Letter)
DOI: 10.1021/ol016361g

Stereoselective 1,2-Additions of α-Alkoxymethyllithiums to Aldehydes

Robert P. Smyj and J. Michael Chong
pp 2903–2906
Publication Date (Web): August 10, 2001 (Letter)
DOI: 10.1021/ol016384v

Tandem Double Intramolecular [4 + 2]/[3 + 2] Cycloadditions of Nitroalkenes

Scott E. Denmark and Laurent Gomez
pp 2907–2910
Publication Date (Web): August 09, 2001 (Letter)
DOI: 10.1021/ol016385n

A Heterocycle-Forming Double Michael Reaction. [5 + 1] Annulation Route to Highly Substituted and Functionalized Piperidines

Freddie Hughes, Jr. and Robert B. Grossman
pp 2911–2914
Publication Date (Web): August 14, 2001 (Letter)
DOI: 10.1021/ol016395o

Effect of Allylic CH3-nFn Groups (n = 1−3) on π-Facial Diastereoselection

Takashi Yamazaki, Tatsuro Ichige, Satoshi Takei, Seiji Kawashita, Tomoya Kitazume, and Toshio Kubota
pp 2915–2918
Publication Date (Web): August 16, 2001 (Letter)
DOI: 10.1021/ol016401g

C-Glycosides to Fused Polycyclic Ethers. An Efficient Entry into the A−D Ring System of Gambierol

Jason M. Cox and Jon D. Rainier
pp 2919–2922
Publication Date (Web): August 08, 2001 (Letter)
DOI: 10.1021/ol016434w

Synthesis of a Broad Array of Highly Functionalized, Enantiomerically Pure Cyclohexanecarboxylic Acid Derivatives by Microbial Dihydroxylation of Benzoic Acid and Subsequent Oxidative and Rearrangement Reactions

Andrew G. Myers, Dionicio R. Siegel, Daniel J. Buzard, and Mark G. Charest
pp 2923–2926
Publication Date (Web): August 17, 2001 (Letter)
DOI: 10.1021/ol010151m

A Synthetic Strategy for the Cyclodepsipeptide Core of the Antitumor Antibiotic Verucopeptin

Karl J. Hale, Linos Lazarides, and Jiaqiang Cai
pp 2927–2930
Publication Date (Web): August 09, 2001 (Letter)
DOI: 10.1021/ol016440s

Novel Polymer-Bound Chiral Selenium Electrophiles

Lars Uehlin and Thomas Wirth
pp 2931–2933
Publication Date (Web): August 10, 2001 (Letter)
DOI: 10.1021/ol0164435

Electrophilic Cyclizations of Vinylcyclopropanols to Tethered Aldehydes

Joo-Hack Youn, Jinhwa Lee, and Jin Kun Cha
pp 2935–2938
Publication Date (Web): August 14, 2001 (Letter)
DOI: 10.1021/ol016490x

Additions and Corrections

N-(tert-Butoxycarbonyl)-N-[4-(dimethylazaniumylidene)-1,4-dihydropyridin-1-ylsulfonyl] Azanide:  A New Sulfamoylating Agent. Structure and Reactivity toward Amines

Jean-Yves Winum, Loic Toupet, Véronique Barragan, Georges Dewynter, and Jean-Louis Montero
p 2939
Publication Date (Web): July 26, 2001 (Additions & Corrections)
DOI: 10.1021/ol010155r

Ethyl(methyl)dioxirane as an Efficient Reagent for the Oxidation of Nucleoside Phosphites into Phosphates under Anhydrous Conditions

Masanori Kataoka, Akira Hattori, Shinya Okino, Mamoru Hyodo, Mitsue Asano, Rie Kawai and Yoshihiro Hayakawa
p 2939
Publication Date (Web): August 01, 2001 (Additions & Corrections)
DOI: 10.1021/ol010160v
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