Table of Contents

Journal Cover
December 13, 2001
Volume 3, Issue 25
Pages 13-4127
For Selected Content:

2001 Division of Organic Chemistry Fellowship Awards

pp 13–17
Publication Date (Web): December 06, 2001 (Letter)
DOI: 10.1021/ol0102491

Letters

Ketone-DNA:  A Versatile Postsynthetic DNA Decoration Platform

Subhakar Dey and Terry L. Sheppard
pp 3983–3986
Publication Date (Web): November 17, 2001 (Letter)
DOI: 10.1021/ol016626r

2-Aryl-2,2-difluoroacetamide FKBP12 Ligands:  Synthesis and X-ray Structural Studies

Gene M. Dubowchik, Vivekananda M. Vrudhula, Bireshwar Dasgupta, Jonathan Ditta, Ti Chen, Steven Sheriff, Karin Sipman, Mark Witmer, Jeffrey Tredup, Dolatrai M. Vyas, Todd A. Verdoorn, Sagarika Bollini, and Alexander Vinitsky
pp 3987–3990
Publication Date (Web): November 17, 2001 (Letter)
DOI: 10.1021/ol0166909

Diastereoselective Addition Reactions of Furyl Aldehydes Using Chiral Boronates as Auxiliary:  Application to the Enantioselective Synthesis of 2,3-Disubstituted Furyl Alcohols

Kin-Fai Chan and Henry N. C. Wong
pp 3991–3994
Publication Date (Web): November 17, 2001 (Letter)
DOI: 10.1021/ol010196n

Efficient Strategy for the Synthesis of Stereopentad Subunits of Scytophycin, Rifamycin S, and Discodermolide

S. BouzBouz and J. Cossy
pp 3995–3998
Publication Date (Web): November 14, 2001 (Letter)
DOI: 10.1021/ol016250h

Cooperative and Selective Lithium Complexation of 2,11,13,22-Tetraaza-5,8,16,19- tetraoxa-1,12-dioxocyclodocosanes

Jau-An Chen, Jun-Liang Lai, Gene Hsiang Lee, Yu Wang, Jen Kuan Su, Hui-Chun Yeh, Wann-Yin Lin, and Man-kit Leung
pp 3999–4002
Publication Date (Web): November 21, 2001 (Letter)
DOI: 10.1021/ol010189z

Intramolecular Palladium(II)-Mediated Alkoxy Carbonylation as a Route to Functionalized Tetrahydropyrans. Synthesis of the C9−C32 Segment of Phorboxazole A

James D. White, Christian L. Kranemann, and Punlop Kuntiyong
pp 4003–4006
Publication Date (Web): November 16, 2001 (Letter)
DOI: 10.1021/ol010193a

Unusual Reagent Control of Diastereoselectivity in the 1,2-Addition of Hard Carbon Nucleophiles to C6-Heteroatom Substituted Cyclohexenones

Harriet A. Lindsay, Catherine L. Salisbury, Wally Cordes, and Matthias C. McIntosh
pp 4007–4010
Publication Date (Web): November 16, 2001 (Letter)
DOI: 10.1021/ol016673j

Enantioselective Synthesis for the Antipodes of Slagenins B and C:  Establishment of Absolute Stereochemistry

Biao Jiang, Jia-Feng Liu, and Sheng-Yin Zhao
pp 4011–4013
Publication Date (Web): November 21, 2001 (Letter)
DOI: 10.1021/ol016689+

Enantiodivergent Synthesis of Either Enantiomer of ABCDE-Ring Analogue of Antitumor Antibiotic Fredericamycin A via Intramolecular [4 + 2] Cycloaddition Approach

Shuji Akai, Toshiaki Tsujino, Nobuhisa Fukuda, Kiyosei Iio, Yoshifumi Takeda, Ken-ichi Kawaguchi, Tadaatsu Naka, Kazuhiro Higuchi, and Yasuyuki Kita
pp 4015–4018
Publication Date (Web): November 16, 2001 (Letter)
DOI: 10.1021/ol016696y

Trehalose-Based Octopus Glycosides for the Synthesis of Carbohydrate-Centered PAMAM Dendrimers and Thiourea-Bridged Glycoclusters

Michael Dubber and Thisbe K. Lindhorst
pp 4019–4022
Publication Date (Web): November 14, 2001 (Letter)
DOI: 10.1021/ol016717o

General Approach for the Synthesis of Sarpagine/Macroline Indole Alkaloids. Enantiospecific Total Synthesis of the Indole Alkaloid Trinervine

Xiaoxiang Liu and James M. Cook
pp 4023–4026
Publication Date (Web): November 16, 2001 (Letter)
DOI: 10.1021/ol0101990

Short Total Syntheses of Both the Putative and Actual Structures of the Clerodane Diterpenoid (±)-Sacacarin by Double Annulation

Robert B. Grossman and Ravindra M. Rasne
pp 4027–4030
Publication Date (Web): November 14, 2001 (Letter)
DOI: 10.1021/ol016748j

Synthesis and Ring-Expanding Oligomerization of an Extremely Strained Macrocyclic Aromatic Ether−Sulfone

Howard M. Colquhoun, Zhixue Zhu, and David J. Williams
pp 4031–4034
Publication Date (Web): November 13, 2001 (Letter)
DOI: 10.1021/ol010201n

Synthesis of 3,4-Disubstituted Isoquinolines via Palladium-Catalyzed Cross-Coupling of o-(1-Alkynyl)benzaldimines and Organic Halides

Guangxiu Dai and Richard C. Larock
pp 4035–4038
Publication Date (Web): November 21, 2001 (Letter)
DOI: 10.1021/ol0102085

Spirocyclic Restriction of Nucleosides. Synthesis of the First Exemplary syn-1-Oxaspiro[4.4]nonanyl Member

Leo A. Paquette, Richard Todd Bibart, Christopher K. Seekamp, and Alexandra L. Kahane
pp 4039–4041
Publication Date (Web): November 10, 2001 (Letter)
DOI: 10.1021/ol010209x

Spirocyclic Restriction of Nucleosides. An Analysis of Protecting Group Feasibility while Accessing Prototype anti-1-Oxaspiro[4.4]nonanyl Mimics

Leo A. Paquette, Dafydd R. Owen, Richard Todd Bibart, and Christopher K. Seekamp
pp 4043–4045
Publication Date (Web): November 10, 2001 (Letter)
DOI: 10.1021/ol010212g

The First Naturally Occurring Tie2 Kinase Inhibitor

Bing-Nan Zhou, Randall K. Johnson, Michael R. Mattern, Paul W. Fisher, and David G. I. Kingston
pp 4047–4049
Publication Date (Web): November 13, 2001 (Letter)
DOI: 10.1021/ol016775+

Novel Conversion of 1,2-Disubstituted cis-Epoxides to One-Carbon Homologated Allylic Alcohols Using Dimethylsulfonium Methylide

Lilian Alcaraz, Andrew Cridland, and Elizabeth Kinchin
pp 4051–4053
Publication Date (Web): November 21, 2001 (Letter)
DOI: 10.1021/ol016782y

Homolytic Carbostannylation of Alkenes and Alkynes with Tributylstannyl Enolates

Katsukiyo Miura, Hiroshi Saito, Naoki Fujisawa, Di Wang, Hisashi Nishikori, and Akira Hosomi
pp 4055–4057
Publication Date (Web): November 20, 2001 (Letter)
DOI: 10.1021/ol016797w

Lactone-Derived Carbon-Centered Radicals:  Formation and Reactivity with Oxygen

Elena V. Bejan, Enrique Font-Sanchis, and J. C. Scaiano
pp 4059–4062
Publication Date (Web): November 16, 2001 (Letter)
DOI: 10.1021/ol0167917

First Generation Design, Synthesis, and Evaluation of Azepine-Based Cryptophycin Analogues

Amos B. Smith, III, Young Shin Cho, Lisa E. Zawacki, Ralph Hirschmann, and George R. Pettit
pp 4063–4066
Publication Date (Web): November 21, 2001 (Letter)
DOI: 10.1021/ol016799g

Visual Recognition of Triamines by Phenolphthalein Derivatives:  Consideration of the Structure of the Colored Complex

Kazunori Tsubaki, Noriyuki Hayashi, Mohammad Nuruzzaman, Tomokazu Kusumoto, and Kaoru Fuji
pp 4067–4069
Publication Date (Web): November 21, 2001 (Letter)
DOI: 10.1021/ol016823q

Visual Enantiomeric Recognition Using Chiral Phenolphthalein Derivatives

Kazunori Tsubaki, Mohammad Nuruzzaman, Tomokazu Kusumoto, Noriyuki Hayashi, Wang Bin-Gui, and Kaoru Fuji
pp 4071–4073
Publication Date (Web): November 21, 2001 (Letter)
DOI: 10.1021/ol016825a

A Stereoselective Synthesis of the C10−C31 (BCDEF Ring) Portion of Pinnatoxin A

Seiichi Nakamura, Jun Inagaki, Tomohiro Sugimoto, Masashi Kudo, Makoto Nakajima, and Shunichi Hashimoto
pp 4075–4078
Publication Date (Web): November 14, 2001 (Letter)
DOI: 10.1021/ol0168364

A Rapid Access to Biaryl Ether Containing Macrocycles by Pairwise Use of Ugi 4CR and Intramolecular SNAr-Based Cycloetherification

Pierre Cristau, Jean-Pierre Vors, and Jieping Zhu
pp 4079–4082
Publication Date (Web): November 10, 2001 (Letter)
DOI: 10.1021/ol0168420

BINOL-Based Diphosphonites as Ligands in the Asymmetric Rh-Catalyzed Conjugate Addition of Arylboronic Acids

Manfred T. Reetz, Dominique Moulin, and Andreas Gosberg
pp 4083–4085
Publication Date (Web): November 16, 2001 (Letter)
DOI: 10.1021/ol010219y

N-Cyclopropylimine-1-pyrroline Rearrangement. A Novel Photochemical Reaction

Pedro J. Campos, Alberto Soldevilla, Diego Sampedro, and Miguel A. Rodríguez
pp 4087–4089
Publication Date (Web): November 16, 2001 (Letter)
DOI: 10.1021/ol016847x

An Intramolecular [2 + 3] Cycloaddition Route to Fused 5-Heterosubstituted Tetrazoles

Zachary P. Demko and K. Barry Sharpless
pp 4091–4094
Publication Date (Web): November 17, 2001 (Letter)
DOI: 10.1021/ol010220x

Generation, Observation, and Free Radical Reactivity of Aliphatic Bisketenes:  The Solution to a Long-Standing Problem

Annette D. Allen, Michael H. Fenwick, Amir Jabri, Huzaifa Rangwala, Kazem Saidi, and Thomas T. Tidwell
pp 4095–4098
Publication Date (Web): November 13, 2001 (Letter)
DOI: 10.1021/ol016853t

Lipase/Palladium-Catalyzed Asymmetric Transformations of Ketoximes to Optically Active Amines

Yoon Kyung Choi, Mi Jung Kim, Yangsoo Ahn, and Mahn-Joo Kim
pp 4099–4101
Publication Date (Web): November 16, 2001 (Letter)
DOI: 10.1021/ol0168622

Palladium-Catalyzed Cross-Coupling Reaction of Triarylbismuths with Aryl Halides and Triflates

Maddali L. N. Rao, Osamu Yamazaki, Shigeru Shimada, Toshifumi Tanaka, Yohichi Suzuki, and Masato Tanaka
pp 4103–4105
Publication Date (Web): November 15, 2001 (Letter)
DOI: 10.1021/ol016885g

Coupling of AlkynylTMS Derivatives with Vinylic Iodides. An Efficient Route to 1,3-Enynes and Dienes

James A. Marshall, Harry R. Chobanian, and Mathew M. Yanik
pp 4107–4110
Publication Date (Web): November 16, 2001 (Letter)
DOI: 10.1021/ol016899m

Efficient Enantioselective Hydrosilylation of Ketones Catalyzed by Air Stable Copper Fluoride−Phosphine Complexes

Sabine Sirol, James Courmarcel, Naouël Mostefai, and Olivier Riant
pp 4111–4113
Publication Date (Web): November 20, 2001 (Letter)
DOI: 10.1021/ol0169170

Chain Extension of Sugar δ-Lactones with the Enolate of tert-Butyl Bromoacetate and Elaboration into Functionalized C-Ketosides, C-Glycosides, and C-Glucosyl Glycines

Frank Schweizer and Toshiyuki Inazu
pp 4115–4118
Publication Date (Web): November 20, 2001 (Letter)
DOI: 10.1021/ol0102343

[2,2]Paracyclophane-Based N,O-Ligands in Alkenylzinc Additions to Aldehydes

Stefan Dahmen and Stefan Bräse
pp 4119–4122
Publication Date (Web): November 20, 2001 (Letter)
DOI: 10.1021/ol016954r

Aerobic Organocatalytic Photoinitiated Arene Oxidations:  Application to Electron Transfer Initiated Cyclization Reactions

V. Satish Kumar, Danielle L. Aubele, and Paul E. Floreancig
pp 4123–4125
Publication Date (Web): November 14, 2001 (Letter)
DOI: 10.1021/ol016996f

Additions and Corrections

Synthesis of Novel Derivatives of 1,4,7-Triazacyclononane

Andrew Warden, Bim Graham, Milton T. W. Hearn, and Leone Spiccia
p 4127
Publication Date (Web): November 15, 2001 (Additions & Corrections)
DOI: 10.1021/ol010256p
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