Synthesis of Target-Specific Radiolabeled Peptides for Diagnostic Imaging

This article is cited by 113 publications.

1. Samad Ahadian, Ramin Banan Sadeghian, Sahar Salehi, Serge Ostrovidov, Hojae Bae, Murugan Ramalingam, and Ali Khademhosseini . Bioconjugated Hydrogels for Tissue Engineering and Regenerative Medicine. Bioconjugate Chemistry 2015, 26 (10) , 1984-2001. https://doi.org/10.1021/acs.bioconjchem.5b00360
2. Flavia Barragán, Paula López-Senín, Luca Salassa, Soledad Betanzos-Lara, Abraha Habtemariam, Virtudes Moreno, Peter J. Sadler, and Vicente Marchán . Photocontrolled DNA Binding of a Receptor-Targeted Organometallic Ruthenium(II) Complex. Journal of the American Chemical Society 2011, 133 (35) , 14098-14108. https://doi.org/10.1021/ja205235m
3. Alessandra Di Cianni, Alfonso Carotenuto, Diego Brancaccio, Ettore Novellino, Jean Claude Reubi, Karin Beetschen, Anna Maria Papini and Mauro Ginanneschi . Novel Octreotide Dicarba-analogues with High Affinity and Different Selectivity for Somatostatin Receptors. Journal of Medicinal Chemistry 2010, 53 (16) , 6188-6197. https://doi.org/10.1021/jm1005868
4. Cara L. Ferreira, Eric Lamsa, Michael Woods, Yin Duan, Pasan Fernando, Corinne Bensimon, Myra Kordos, Katharina Guenther, Paul Jurek and Garry E. Kiefer . Evaluation of Bifunctional Chelates for the Development of Gallium-Based Radiopharmaceuticals. Bioconjugate Chemistry 2010, 21 (3) , 531-536. https://doi.org/10.1021/bc900443a
5. Xin Sheng, Xun Guo, Xiao-Min Lu, Guo-Yuan Lu, Ying Shao, Fang Liu and Qiang Xu . DNA Binding, Cleavage, and Cytotoxic Activity of the Preorganized Dinuclear Zinc(II) Complex of Triazacyclononane Derivatives. Bioconjugate Chemistry 2008, 19 (2) , 490-498. https://doi.org/10.1021/bc700322w
6. Luis M. De León-Rodríguez and Zoltan Kovacs . The Synthesis and Chelation Chemistry of DOTA−Peptide Conjugates. Bioconjugate Chemistry 2008, 19 (2) , 391-402. https://doi.org/10.1021/bc700328s
7. Debora D’Addona, Alfonso Carotenuto, Ettore Novellino, Véronique Piccand, Jean Claude Reubi, Alessandra Di Cianni, Francesca Gori, Anna Maria Papini and Mauro Ginanneschi. Novel sst5-Selective Somatostatin Dicarba-Analogues: Synthesis and Conformation−Affinity Relationships. Journal of Medicinal Chemistry 2008, 51 (3) , 512-520. https://doi.org/10.1021/jm070886i
8. Simonetta Geninatti Crich,, Claudia Cabella,, Alessandro Barge,, Simona Belfiore,, Cristina Ghirelli,, Luciano Lattuada,, Stefania Lanzardo,, Armando Mortillaro,, Lorenzo Tei,, Massimo Visigalli,, Guido Forni, and, Silvio Aime. In Vitro and in Vivo Magnetic Resonance Detection of Tumor Cells by Targeting Glutamine Transporters with Gd-Based Probes. Journal of Medicinal Chemistry 2006, 49 (16) , 4926-4936. https://doi.org/10.1021/jm0601093
9. Lassi Jaakkola,, Alice Ylikoski, and, Jari Hovinen. Simple Synthesis of a Building Block for Solid-Phase Labeling of Oligonucleotides with 1,4,7,10-Tetraazacyclododecane-1,4,7,10-tetraacetic Acid (DOTA). Bioconjugate Chemistry 2006, 17 (4) , 1105-1107. https://doi.org/10.1021/bc0600362
10. Jari Peuralahti,, Lassi Jaakkola,, Veli-Matti Mukkala, and, Jari Hovinen. Synthesis of Building Blocks for Solid-Phase Introduction of Diethylenetriaminepentaacetic Acid (DTPA) to Oligonucleotides and Oligopeptides. Bioconjugate Chemistry 2006, 17 (3) , 855-859. https://doi.org/10.1021/bc0503667
11. Young Soo Chang,, Jae Min Jeong,, Yun-Sang Lee,, Hyung Woo Kim,, Ganesha B. Rai,, Seung Jin Lee,, Dong Soo Lee,, June-Key Chung, and, Myung Chul Lee. Preparation of 18F-Human Serum Albumin:  A Simple and Efficient Protein Labeling Method with 18F Using a Hydrazone-Formation Method. Bioconjugate Chemistry 2005, 16 (5) , 1329-1333. https://doi.org/10.1021/bc050086r
12. William E. P. Greenland and, Philip J. Blower. Water-Soluble Phosphines for Direct Labeling of Peptides with Technetium and Rhenium:  Insights from Electrospray Mass Spectrometry. Bioconjugate Chemistry 2005, 16 (4) , 939-948. https://doi.org/10.1021/bc0500600
13. Roberta Visentin,, Gianfranco Pasut,, Francesco Maria Veronese, and, Ulderico Mazzi. Highly Efficient Technetium-99m Labeling Procedure Based on the Conjugation of N-[N-(3-Diphenylphosphinopropionyl)glycyl]cysteine Ligand with Poly(ethylene glycol). Bioconjugate Chemistry 2004, 15 (5) , 1046-1054. https://doi.org/10.1021/bc049896d
14. Wen-Yuan Hsieh and, Shuang Liu. Synthesis, Characterization, and Structures of Indium In(DTPA-BA2) and Yttrium Y(DTPA-BA2)(CH3OH) Complexes (BA = Benzylamine):  Models for 111In- and 90Y-Labeled DTPA-Biomolecule Conjugates. Inorganic Chemistry 2004, 43 (19) , 6006-6014. https://doi.org/10.1021/ic049973g
15. David C. Onthank,, Shuang Liu,, Paula J. Silva,, John A. Barrett,, Thomas D. Harris,, Simon P. Robinson, and, D. Scott Edwards. 90Y and 111In Complexes of a DOTA-Conjugated Integrin αvβ3 Receptor Antagonist:  Different but Biologically Equivalent. Bioconjugate Chemistry 2004, 15 (2) , 235-241. https://doi.org/10.1021/bc034108q
16. Shuang Liu,, Zhengjie He,, Wen-Yuan Hsieh, and, Phillip E. Fanwick. Synthesis, Characterization, and X-ray Crystal Structure of In(DOTA-AA) (AA = p-Aminoanilide):  A Model for 111In-Labeled DOTA-Biomolecule Conjugates. Inorganic Chemistry 2003, 42 (26) , 8831-8837. https://doi.org/10.1021/ic0349914
17. Tatsushi Toyokuni,, Joseph C. Walsh,, Alan Dominguez,, Michael E. Phelps,, Jorge R. Barrio,, Sanjiv S. Gambhir, and, Nagichettiar Satyamurthy. Synthesis of a New Heterobifunctional Linker, N-[4-(Aminooxy)butyl]maleimide, for Facile Access to a Thiol-Reactive 18F-Labeling Agent. Bioconjugate Chemistry 2003, 14 (6) , 1253-1259. https://doi.org/10.1021/bc034107y
18. Shuang Liu,, Charlie E. Ellars, and, D. Scott Edwards. Ascorbic Acid:  Useful as a Buffer Agent and Radiolytic Stabilizer for Metalloradiopharmaceuticals. Bioconjugate Chemistry 2003, 14 (5) , 1052-1056. https://doi.org/10.1021/bc034109i
19. György Trencsényi, Zita Képes. Scandium-44: Diagnostic Feasibility in Tumor-Related Angiogenesis. International Journal of Molecular Sciences 2023, 24 (8) , 7400. https://doi.org/10.3390/ijms24087400
20. Hendris Wongso. Natural product-based radiopharmaceuticals: Focus on curcumin and its analogs, flavonoids, and marine peptides. Journal of Pharmaceutical Analysis 2022, 12 (3) , 380-393. https://doi.org/10.1016/j.jpha.2021.07.006
21. Subhani M. Okarvi, Ibrahim Al-Jammaz. Synthesis, Radiolabeling, and Preclinical Evaluation of 68 Ga/ 177 Lu-Labeled Leuprolide Peptide Analog for the Detection of Breast Cancer. Cancer Biotherapy and Radiopharmaceuticals 2022, 37 (5) , 372-383. https://doi.org/10.1089/cbr.2021.0370
22. Andrew J. Hall, Mohammad B. Haskali. Radiolabelled Peptides: Optimal Candidates for Theranostic Application in Oncology. Australian Journal of Chemistry 2022, 75 (2) , 34-54. https://doi.org/10.1071/CH21118
23. Khurram Shahzad, Aman Shah Abdul Majid, Mumtaz Khan, Muhammad Adnan Iqbal, Asjad Ali. Recent advances in the synthesis of ( 99m Technetium) based radio-pharmaceuticals. Reviews in Inorganic Chemistry 2021, 41 (3) , 151-198. https://doi.org/10.1515/revic-2020-0021
24. Crhisterra Ellen Kusumaningrum, Eva Maria Widyasari, Maula Eka Sriyani, Hendris Wongso. Pharmacological activities and potential use of bovine colostrum for peptide-based radiopharmaceuticals: A review. Pharmacia 2021, 68 (2) , 471-477. https://doi.org/10.3897/pharmacia.68.e65537
25. Sajjad Ahmadpour, Seyed Jalal Hosseinimehr. Recent developments in peptide-based SPECT radiopharmaceuticals for breast tumor targeting. Life Sciences 2019, 239 , 116870. https://doi.org/10.1016/j.lfs.2019.116870
26. Andrea Caporale, Cristina Bolzati, Giuseppina Maria Incisivo, Nicola Salvarese, Paolo Grieco, Menotti Ruvo. Improved synthesis on solid phase of dithiocarbamic cRGD ‐derivative and 99m Tc ‐radiolabelling. Journal of Peptide Science 2019, 25 (2) https://doi.org/10.1002/psc.3140
27. Chiara Testa, Debora D'Addona, Mario Scrima, Anna Maria Tedeschi, Anna Maria D'Ursi, Claire Bernhard, Franck Denat, Claudia Bello, Paolo Rovero, Michael Chorev, Anna Maria Papini. Design, synthesis, and conformational studies of [DOTA]‐Octreotide analogs containing [1,2,3]triazolyl as a disulfide mimetic. Peptide Science 2018, 110 (5) https://doi.org/10.1002/pep2.24071
28. Feng Gao, Wiebke Sihver, Ralf Bergmann, Birgit Belter, Cristina Bolzati, Nicola Salvarese, Jörg Steinbach, Jens Pietzsch, Hans‐Jürgen Pietzsch. Synthesis, Characterization, and Initial Biological Evaluation of [ 99m Tc]Tc‐Tricarbonyl‐labeled DPA‐α‐MSH Peptide Derivatives for Potential Melanoma Imaging. ChemMedChem 2018, 13 (11) , 1146-1158. https://doi.org/10.1002/cmdc.201800110
29. Syed Qaiser Shah, Samia Mahmood. Evaluation of 99m Tc-Labeled Bevacizumab– N- HYNIC Conjugate in Human Ovarian Tumor Xenografts. Cancer Biotherapy and Radiopharmaceuticals 2018, 33 (3) , 96-102. https://doi.org/10.1089/cbr.2017.2323
30. Pauline Désogère, Luis F. Tapias, Tyson A. Rietz, Nicholas Rotile, Francesco Blasi, Helen Day, Justin Elliott, Bryan C. Fuchs, Michael Lanuti, Peter Caravan. Optimization of a Collagen-Targeted PET Probe for Molecular Imaging of Pulmonary Fibrosis. Journal of Nuclear Medicine 2017, 58 (12) , 1991-1996. https://doi.org/10.2967/jnumed.117.193532
31. Ryota Yoshida, Katsuhiro Isozaki, Tomoya Yokoi, Nobuhiro Yasuda, Koichiro Sadakane, Takahiro Iwamoto, Hikaru Takaya, Masaharu Nakamura. ONO-pincer ruthenium complex-bound norvaline for efficient catalytic oxidation of methoxybenzenes with hydrogen peroxide. Organic & Biomolecular Chemistry 2016, 14 (31) , 7468-7479. https://doi.org/10.1039/C6OB00969G
32. Sadaaki Kimura, Yuu Kakishima, Takahiro Kuchimaru, Shinae Kizaka-Kondoh, Mitsuyoshi Yoshimoto, Hirofumi Fujii, Izumi O. Umeda. Application of HaloTag® Technology to in Vivo Molecular Imaging Using Protein Probes Labeled by Metallic Radionuclides. RADIOISOTOPES 2016, 65 (6) , 247-255. https://doi.org/10.3769/radioisotopes.65.247
33. Julie K. Jang, David Canter, Peisheng Hu, Alan L. Epstein, Leslie A. Khawli. Labeling and Imaging Techniques for Quantification of Therapeutic Biologics. 2015, 1-24. https://doi.org/10.1002/9780470571224.pse554
34. Eric W. Price, Chris Orvig. The Chemistry of Inorganic Nuclides ( 86 Y, 68 Ga, 64 Cu, 89 Zr, 124 I). 2014, 105-135. https://doi.org/10.1002/9781118854754.ch5
35. Prakash Sista, Koushik Ghosh, Jennifer S. Martinez, Reginaldo C. Rocha. Metallo-Biopolymers: Conjugation Strategies and Applications. Polymer Reviews 2014, 54 (4) , 627-676. https://doi.org/10.1080/15583724.2014.913063
36. Ella Kriemen, Erik Ruf, Ulrich Behrens, Wolfgang Maison. Synthesis of 1,4,7,10‐Tetra‐azacyclododecan‐1,4,7,10‐tetra‐azidoethylacetic Acid (DOTAZA) and Related “Clickable” DOTA Derivatives. Chemistry – An Asian Journal 2014, 9 (8) , 2197-2204. https://doi.org/10.1002/asia.201402250
37. Grant Sugiura, Helen Kühn, Max Sauter, Uwe Haberkorn, Walter Mier. Radiolabeling Strategies for Tumor-Targeting Proteinaceous Drugs. Molecules 2014, 19 (2) , 2135-2165. https://doi.org/10.3390/molecules19022135
38. Eric W. Price, Chris Orvig. Matching chelators to radiometals for radiopharmaceuticals. Chem. Soc. Rev. 2014, 43 (1) , 260-290. https://doi.org/10.1039/C3CS60304K
39. Efrosyni Themistou, Giuseppe Battaglia, Steven P. Armes. Facile synthesis of thiol-functionalized amphiphilic polylactide–methacrylic diblock copolymers. Polym. Chem. 2014, 5 (4) , 1405-1417. https://doi.org/10.1039/C3PY01446K
40. Qaisar Nadeem, Daniel Can, Yunjun Shen, Michael Felber, Zaid Mahmood, Roger Alberto. Synthesis of tripeptide derivatized cyclopentadienyl complexes of technetium and rhenium as radiopharmaceutical probes. Organic & Biomolecular Chemistry 2014, 12 (12) , 1966. https://doi.org/10.1039/c3ob41866a
41. Kazuki Ogata, Daisuke Sasano, Tomoya Yokoi, Katsuhiro Isozaki, Ryota Yoshida, Toshio Takenaka, Hirofumi Seike, Tetsuya Ogawa, Hiroki Kurata, Nobuhiro Yasuda, Hikaru Takaya, Masaharu Nakamura. Synthesis and Self‐Assembly of NCN‐Pincer Pd‐Complex‐Bound Norvalines. Chemistry – A European Journal 2013, 19 (37) , 12356-12375. https://doi.org/10.1002/chem.201301513
42. Mazen Jamous, Uwe Haberkorn, Walter Mier. Synthesis of Peptide Radiopharmaceuticals for the Therapy and Diagnosis of Tumor Diseases. Molecules 2013, 18 (3) , 3379-3409. https://doi.org/10.3390/molecules18033379
43. Pauline Désogère, Claire Bernhard, Christine Goze, Marie‐José Penouilh, Yoann Rousselin, Franck Denat. Selectively Functionalized Constrained Polyazamacrocycles: Building Blocks for Multifunctional Chelating Agents. European Journal of Organic Chemistry 2013, 2013 (8) , 1538-1545. https://doi.org/10.1002/ejoc.201201337
44. S. M. Okarvi, H. R. Maecke. Peptides for Nuclear Medicine Therapy: Chemical Properties and Production. 2013, 105-123. https://doi.org/10.1007/174_2013_921
45. Raunak Varshney, Puja P. Hazari, P. Fernandez, J. Schulz, M. Allard, Anil K. Mishra. 68Ga-Labeled Bombesin Analogs for Receptor-Mediated Imaging. 2013, 221-256. https://doi.org/10.1007/978-3-642-27994-2_12
46. Katsuhiro Isozaki, Yusuke Haga, Kazuki Ogata, Takeshi Naota, Hikaru Takaya. Metal array fabrication based on ultrasound-induced self-assembly of metalated dipeptides. Dalton Transactions 2013, 42 (45) , 15953. https://doi.org/10.1039/c3dt51696b
47. Claire Bernhard, Mathieu Moreau, Damien Lhenry, Christine Goze, Frédéric Boschetti, Yoann Rousselin, François Brunotte, Franck Denat. DOTAGA–Anhydride: A Valuable Building Block for the Preparation of DOTA‐Like Chelating Agents. Chemistry – A European Journal 2012, 18 (25) , 7834-7841. https://doi.org/10.1002/chem.201200132
48. Leonardo Manzoni, Laura Belvisi, Daniela Arosio, Maria Paola Bartolomeo, Aldo Bianchi, Chiara Brioschi, Federica Buonsanti, Claudia Cabella, Cesare Casagrande, Monica Civera, Marilenia De Matteo, Lorenza Fugazza, Luciano Lattuada, Federico Maisano, Luigi Miragoli, Cristina Neira, Michael Pilkington‐Miksa, Carlo Scolastico. Synthesis of Gd and 68 Ga Complexes in Conjugation with a Conformationally Optimized RGD Sequence as Potential MRI and PET Tumor‐Imaging Probes. ChemMedChem 2012, 7 (6) , 1084-1093. https://doi.org/10.1002/cmdc.201200043
49. Yun-Sang Lee, Jae Min Jeong. Inorganic Radionuclides for Nuclear Medicine Therapy. 2012, 151-163. https://doi.org/10.1007/174_2012_704
50. Susan Roosenburg, Peter Laverman, Floris L. van Delft, Otto C. Boerman. Radiolabeled CCK/gastrin peptides for imaging and therapy of CCK2 receptor-expressing tumors. Amino Acids 2011, 41 (5) , 1049-1058. https://doi.org/10.1007/s00726-010-0501-y
51. Eva Balentova, Charlotte Collet, Sandrine Lamandé-Langle, Françoise Chrétien, David Thonon, Joël Aerts, Christian Lemaire, André Luxen, Yves Chapleur. Synthesis and hydrolytic stability of novel 3-[18F]fluoroethoxybis(1-methylethyl)silyl]propanamine-based prosthetic groups. Journal of Fluorine Chemistry 2011, 132 (4) , 250-257. https://doi.org/10.1016/j.jfluchem.2011.01.011
52. Roger Alberto. Metal‐Based Radiopharmaceuticals. 2011, 253-282. https://doi.org/10.1002/9783527633104.ch9
53. R. Alberto, U. Abram. 99mTc: Labeling Chemistry and Labeled Compounds. 2011, 2073-2120. https://doi.org/10.1007/978-1-4419-0720-2_43
54. M. Fani, S. Good, H. R. Maecke. Radiometals (non-Tc, non-Re) and Bifunctional Labeling Chemistry. 2011, 2143-2178. https://doi.org/10.1007/978-1-4419-0720-2_45
55. Rodrigo Teodoro, Bluma Linkowski Faintuch, Eutimio Gustavo Fernández Núñez, Rodrigo Guimarães Queiróz. Neurotensin(8–13) analogue: radiolabeling and biological evaluation using different chelators. Nuclear Medicine and Biology 2011, 38 (1) , 113-120. https://doi.org/10.1016/j.nucmedbio.2010.06.011
56. Luciano Lattuada, Alessandro Barge, Giancarlo Cravotto, Giovanni Battista Giovenzana, Lorenzo Tei. The synthesis and application of polyamino polycarboxylic bifunctional chelating agents. Chemical Society Reviews 2011, 40 (5) , 3019. https://doi.org/10.1039/c0cs00199f
57. João D. G. Correia, António Paulo, Paula D. Raposinho, Isabel Santos. Radiometallated peptides for molecular imaging and targeted therapy. Dalton Transactions 2011, 40 (23) , 6144. https://doi.org/10.1039/c0dt01599g
58. Dinesh Shetty, Yun-Sang Lee, Jae Min Jeong. 68Ga-Labeled Radiopharmaceuticals for Positron Emission Tomography. Nuclear Medicine and Molecular Imaging 2010, 44 (4) , 233-240. https://doi.org/10.1007/s13139-010-0056-6
59. Susanne Bomke, Michael Sperling, Uwe Karst. Organometallic derivatizing agents in bioanalysis. Analytical and Bioanalytical Chemistry 2010, 397 (8) , 3483-3494. https://doi.org/10.1007/s00216-010-3611-1
60. Catherine Cote, Rein U. Kirss. Rhenium tricarbonyl complexes of 1-benzyl-4-(5-bipyridyl)-1H-1,2,3-triazoles. Inorganica Chimica Acta 2010, 363 (11) , 2520-2525. https://doi.org/10.1016/j.ica.2010.04.019
61. Raymond M. Reilly. The Radiochemistry of Monoclonal Antibodies and Peptides. 2010, 39-100. https://doi.org/10.1002/9780470613214.ch2
62. Levente K. Meszaros, Anica Dose, Stefano C.G. Biagini, Philip J. Blower. Hydrazinonicotinic acid (HYNIC) – Coordination chemistry and applications in radiopharmaceutical chemistry. Inorganica Chimica Acta 2010, 363 (6) , 1059-1069. https://doi.org/10.1016/j.ica.2010.01.009
63. Raymond M. Reilly. The Radiopharmaceutical Science of Monoclonal Antibodies and Peptides for Imaging and Targeted In Situ Radiotherapy of Malignancies. 2010, 1-60. https://doi.org/10.1002/9780470571224.pse318
64. Corinne Bensimon, Russell Redshaw. Antibody Radiolabeling. 2010, 323-344. https://doi.org/10.1007/978-0-387-76643-0_19
65. N. Sadeghzadeh, M. Gandomkar, R. Najafi, M. Shafiei, S. E. Sadat Ebrahimi, A. Shafiee, B. Larijani. Preparation and evaluation of a new 99mTc labeled bombesin derivative for tumor imaging. Journal of Radioanalytical and Nuclear Chemistry 2010, 283 (1) , 181-187. https://doi.org/10.1007/s10967-009-0138-z
66. Giuseppe Gugliotta, Mauro Botta, Lorenzo Tei. AAZTA-based bifunctional chelating agents for the synthesis of multimeric/dendrimeric MRI contrast agents. Organic & Biomolecular Chemistry 2010, 8 (20) , 4569. https://doi.org/10.1039/c0ob00096e
67. Ghassan Bechara, Nadine Leygue, Chantal Galaup, Béatrice Mestre, Claude Picard. An efficient route to pyridine and 2,2′-bipyridine macrocycles incorporating a triethylenetetraminetetraacetic acid core as ligand for lanthanide ions. Tetrahedron Letters 2009, 50 (47) , 6522-6525. https://doi.org/10.1016/j.tetlet.2009.09.030
68. Rafael Torres Martin de Rosales, Erik Årstad, Philip J. Blower. Nuclear imaging of molecular processes in cancer. Targeted Oncology 2009, 4 (3) , 183-197. https://doi.org/10.1007/s11523-009-0120-2
69. . Chemistry of Metal Radionuclides (Rb, Ga, In, Y, Cu and Tc). 2009, 179-196. https://doi.org/10.1007/978-3-540-76735-0_12
70. Michaela Försterová, Miloš Petřík, Alice Lázničková, Milan Lázníček, Petr Hermann, Ivan Lukeš, František Melichar. Complexation and biodistribution study of 111In and 90Y complexes of bifunctional phosphinic acid analogs of H4dota. Applied Radiation and Isotopes 2009, 67 (1) , 21-29. https://doi.org/10.1016/j.apradiso.2008.08.013
71. Sara Lacerda, M. Paula Campello, Fernanda Marques, Lurdes Gano, Vojtěch Kubíček, Petra Fousková, Éva Tóth, Isabel Santos. A novel tetraazamacrocycle bearing a thiol pendant arm for labeling biomolecules with radiolanthanides. Dalton Transactions 2009, 60 (23) , 4509. https://doi.org/10.1039/b820375j
72. Hancheng Cai, John Fissekis, Peter S. Conti. Synthesis of a novel bifunctional chelator AmBaSar based on sarcophagine for peptide conjugation and 64Cu radiolabelling. Dalton Transactions 2009, 17 (27) , 5395. https://doi.org/10.1039/b902210d
73. Alessandro Barge, Enrico Cappelletti, Giancarlo Cravotto, Aurelia Ferrigato, Luciano Lattuada, Fabio Marinoni, Lorenzo Tei. Synthesis of functionalised HP-DO3A chelating agents for conjugation to biomolecules. Organic & Biomolecular Chemistry 2009, 7 (18) , 3810. https://doi.org/10.1039/b905369g
74. Lorenzo Tei, Giuseppe Gugliotta, Stefano Avedano, Giovanni B. Giovenzana, Mauro Botta. Application of the Ugi four-component reaction to the synthesis of ditopic bifunctional chelating agents. Organic & Biomolecular Chemistry 2009, 7 (21) , 4406. https://doi.org/10.1039/b907932g
75. Flavia Barragán, Virtudes Moreno, Vicente Marchán. Solid-phase synthesis and DNA binding studies of dichloroplatinum(ii) conjugates of dicarba analogues of octreotide as new anticancer drugs. Chemical Communications 2009, 99 (31) , 4705. https://doi.org/10.1039/b909698a
76. Cornelia Walther, Ingo Ott, Ronald Gust, Ines Neundorf. Specific labeling with potent radiolabels alters the uptake of cell‐penetrating peptides. Peptide Science 2009, 92 (5) , 445-451. https://doi.org/10.1002/bip.21218
77. Shuang Liu. Bifunctional coupling agents for radiolabeling of biomolecules and target-specific delivery of metallic radionuclides. Advanced Drug Delivery Reviews 2008, 60 (12) , 1347-1370. https://doi.org/10.1016/j.addr.2008.04.006
78. Michaela Försterová, Zuzana Jandurová, Fernanda Marques, Lurdes Gano, Přemysl Lubal, Jakub Vaněk, Petr Hermann, Isabel Santos. Chemical and biological evaluation of 153Sm and 166Ho complexes of 1,4,7,10-tetraazacyclododecane-1,4,7,10-tetrakis(methylphosphonic acid monoethylester) (H4dotpOEt). Journal of Inorganic Biochemistry 2008, 102 (7) , 1531-1540. https://doi.org/10.1016/j.jinorgbio.2008.02.002
79. Georg Dirscherl, Burkhard König. The Use of Solid‐Phase Synthesis Techniques for the Preparation of Peptide–Metal Complex Conjugates. European Journal of Organic Chemistry 2008, 2008 (4) , 597-634. https://doi.org/10.1002/ejoc.200700787
80. Pritesh Patel, Phil Jones, Richard Handy, Chris Harrington, Peter Marshall, E. Hywel Evans. Isotopic labelling of peptides and isotope ratio analysis using LC–ICP–MS: a preliminary study. Analytical and Bioanalytical Chemistry 2008, 390 (1) , 61-65. https://doi.org/10.1007/s00216-007-1432-7
81. Miguel A. Avila-Rodriguez, Jonathon A. Nye, Robert J. Nickles. Production and separation of non-carrier-added 86Y from enriched 86Sr targets. Applied Radiation and Isotopes 2008, 66 (1) , 9-13. https://doi.org/10.1016/j.apradiso.2007.07.027
82. Xin Sheng, Xiao‐Min Lu, Yue‐Ting Chen, Guo‐Yuan Lu, Jing‐Jing Zhang, Ying Shao, Fang Liu, Qiang Xu. Synthesis, DNA‐Binding, Cleavage, and Cytotoxic Activity of New 1,7‐Dioxa‐4,10‐diazacyclododecane Artificial Receptors Containing Bisguanidinoethyl or Diaminoethyl Double Side Arms. Chemistry – A European Journal 2007, 13 (34) , 9703-9712. https://doi.org/10.1002/chem.200700549
83. Ying Li, Xiao-Min Lu, Xin Sheng, Guo-Yuan Lu, Ying Shao, Qiang Xu. DNA cleavage promoted by Cu2+ complex of cyclen containing pyridine subunit. Journal of Inclusion Phenomena and Macrocyclic Chemistry 2007, 59 (1-2) , 91-98. https://doi.org/10.1007/s10847-007-9299-y
84. Sebastian Knör, Armin Modlinger, Thorsten Poethko, Margret Schottelius, Hans‐Jürgen Wester, Horst Kessler. Synthesis of Novel 1,4,7,10‐Tetraazacyclodecane‐1,4,7,10‐Tetraacetic Acid (DOTA) Derivatives for Chemoselective Attachment to Unprotected Polyfunctionalized Compounds. Chemistry – A European Journal 2007, 13 (21) , 6082-6090. https://doi.org/10.1002/chem.200700231
85. Stefania Agostini, Cristina Bolzati, Eliana Didonè, Mario Cavazza‐Ceccato, Fiorenzo Refosco, Luigi Aloj, Claudio Arra, Michela Aurilio, Anna Lucia Tornesello, Diego Tesauro, Giancarlo Morelli. The [Tc(N)(PNP)] 2+ metal fragment labeled cholecystokinin‐8 (CCK8) peptide for CCK‐2 receptors imaging: in vitro and in vivo studies. Journal of Peptide Science 2007, 13 (4) , 211-219. https://doi.org/10.1002/psc.834
86. Alessandro Barge, Giancarlo Cravotto, Bruna Robaldo, Eliana Gianolio, Silvio Aime. New CD derivatives as self-assembling contrast agents for magnetic resonance imaging (MRI). Journal of Inclusion Phenomena and Macrocyclic Chemistry 2007, 57 (1-4) , 489-495. https://doi.org/10.1007/s10847-006-9239-2
87. Dominik Heckmann, Horst Kessler. Design and Chemical Synthesis of Integrin Ligands. 2007, 463-503. https://doi.org/10.1016/S0076-6879(07)26020-3
88. Rita Delgado, Vítor Félix, Luís M. P. Lima, David W. Price. Metal complexes of cyclen and cyclam derivatives useful for medical applications: a discussion based on thermodynamic stability constants and structural data. Dalton Trans. 2007, 99 (26) , 2734-2745. https://doi.org/10.1039/B704360K
89. Byunghee Yoo, Mark D. Pagel. A facile synthesis of α-amino-DOTA as a versatile molecular imaging probe. Tetrahedron Letters 2006, 47 (41) , 7327-7330. https://doi.org/10.1016/j.tetlet.2006.08.019
90. Jari Peuralahti, Liisa Meriö, Veli-Matti Mukkala, Kaj Blomberg, Jari Hovinen. Synthesis and properties of a neutral derivative of diethylenetriaminepentaacetic acid (DTPA). Bioorganic & Medicinal Chemistry Letters 2006, 16 (18) , 4760-4762. https://doi.org/10.1016/j.bmcl.2006.06.088
91. Luciano Lattuada, Silvia Demattio, Veronica Vincenzi, Claudia Cabella, Massimo Visigalli, Silvio Aime, Simonetta Geninatti Crich, Eliana Gianolio. Magnetic resonance imaging of tumor cells by targeting the amino acid transport system. Bioorganic & Medicinal Chemistry Letters 2006, 16 (15) , 4111-4114. https://doi.org/10.1016/j.bmcl.2006.04.081
92. Julien Le Gal, Sandra Michaud, Marie Gressier, Yvon Coulais, Eric Benoist. Synthesis, metal complexation and biological evaluation of a novel semi-rigid bifunctional chelating agent for 99mTc labelling. Bioorganic & Medicinal Chemistry 2006, 14 (9) , 2904-2909. https://doi.org/10.1016/j.bmc.2005.12.005
93. Shu-Hui Wan, Feng Liang, Xiao-Qin Xiong, Li Yang, Xiao-Jun Wu, Ping Wang, Xiang Zhou, Cheng-Tai Wu. DNA hydrolysis promoted by 1,7-dimethyl-1,4,7,10-tetraazacyclododecane. Bioorganic & Medicinal Chemistry Letters 2006, 16 (10) , 2804-2806. https://doi.org/10.1016/j.bmcl.2006.01.106
94. Daniela Arosio, Matteo Bertoli, Leonardo Manzoni, Carlo Scolastico. Click chemistry to functionalise peptidomimetics. Tetrahedron Letters 2006, 47 (22) , 3697-3700. https://doi.org/10.1016/j.tetlet.2006.03.149
95. Jari Hovinen. Synthesis of Aminooxy‐Functionalized Lanthanide(III) Chelates for Carbonyl‐Group Conjugation. Chemistry & Biodiversity 2006, 3 (3) , 296-303. https://doi.org/10.1002/cbdv.200690032
96. Subhani M. Okarvi, Ibrahim A. Jammaz. Preparation and In Vitro and In Vivo Evaluation of Technetium- 99m -Labeled Folate and Methotrexate Conjugates as Tumor Imaging Agents. Cancer Biotherapy and Radiopharmaceuticals 2006, 21 (1) , 49-60. https://doi.org/10.1089/cbr.2006.21.49
97. Matthew S. Tremblay, Dalibor Sames. Synthesis of luminescent heterometallic bis-lanthanide complexes via selective, sequential metallation. Chemical Communications 2006, 102 (39) , 4116. https://doi.org/10.1039/b607949k
98. Karin A Stephenson, Sangeeta Ray Banerjee, Nicole McFarlane, Douglas R Boreham, Kevin P Maresca, John W Babich, Jon Zubieta, John F Valliant. A convenient solid-phase synthesis methodology for preparing peptide-derived molecular imaging agents Synthesis, characterization, and in vitro screening of Tc(I) chemotactic peptide conjugates. Canadian Journal of Chemistry 2005, 83 (12) , 2060-2066. https://doi.org/10.1139/v05-224
99. Luciano Lattuada, Milena Gabellini. Straightforward Synthesis of a Novel Maleimide‐DTPA Bifunctional Chelating Agent. Synthetic Communications 2005, 35 (18) , 2409-2413. https://doi.org/10.1080/00397910500189569
100. Bhupender S. Chhikara, Nitin Kumar, Vibha Tandon, Anil K. Mishra. Synthesis and evaluation of bifunctional chelating agents derived from bis(2-aminophenylthio)alkane for radioimaging with 99mTc. Bioorganic & Medicinal Chemistry 2005, 13 (15) , 4713-4720. https://doi.org/10.1016/j.bmc.2005.04.073