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Histamine H3 Receptor as a Drug Discovery Target

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Chemical Research, Merck Research Laboratories, 2015 Galloping Hill Road, Kenilworth, New Jersey 07033, United States
*To whom correspondence should be addressed. Phone: 1-908-740-3909. Fax: 1-908-740-7152. E-mail: [email protected]
Cite this: J. Med. Chem. 2011, 54, 1, 26–53
Publication Date (Web):November 9, 2010
Copyright © 2010 American Chemical Society

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    Details of the H3 receptor signaling pathways (summarized in Figure 4) and details of the clinical trials targeting H3 receptor (as listed on This material is available free of charge via the Internet at

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