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Designing synthetic superagonists of C3a anaphylatoxin

Cite this: Biochemistry 1991, 30, 15, 3603–3612
Publication Date (Print):April 16, 1991
https://doi.org/10.1021/bi00229a003
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    23. Andreas Klos, Elisabeth Wende, Kathryn J. Wareham, Peter N. Monk. International Union of Basic and Clinical Pharmacology. LXXXVII. Complement Peptide C5a, C4a, and C3a Receptors. Pharmacological Reviews 2013, 65 (1) , 500-543. https://doi.org/10.1124/pr.111.005223
    24. Sakeen W. Kashem, Hariharan Subramanian, Sarah J. Collington, Paola Magotti, John D. Lambris, Hydar Ali. G protein coupled receptor specificity for C3a and compound 48/80-induced degranulation in human mast cells: Roles of Mas-related genes MrgX1 and MrgX2. European Journal of Pharmacology 2011, 668 (1-2) , 299-304. https://doi.org/10.1016/j.ejphar.2011.06.027
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    29. Jinming Gao, Hyeryun Choe, Dalena Bota, Paulette L. Wright, Craig Gerard, Norma P. Gerard. Sulfation of Tyrosine 174 in the Human C3a Receptor Is Essential for Binding of C3a Anaphylatoxin. Journal of Biological Chemistry 2003, 278 (39) , 37902-37908. https://doi.org/10.1074/jbc.M306061200
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