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Conformationally Restricted Competitive Antagonists of Human/Rat Corticotropin-Releasing Factor

Cite this: J. Med. Chem. 1994, 37, 10, 1450–1459
Publication Date (Print):May 1, 1994
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    This article is cited by 57 publications.

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    42. K. Eckart, O. Jahn, J. Radulovic, M. Radulovic, T. Blank, O. Stiedl, O. Brauns, H. Tezval, T. Zeyda, J. Spiess. Pharmacology and Biology of Corticotropin-Releasing Factor (CRF) Receptors. Receptors and Channels 2002, 8 (3-4) , 163-177.
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    50. Andreas Rühmann, Ines Bonk, Chijen R. Lin, Michael G. Rosenfeld, Joachim Spiess. Structural requirements for peptidic antagonists of the corticotropin-releasing factor receptor (CRFR): Development of CRFR2β-selective antisauvagine-30. Proceedings of the National Academy of Sciences 1998, 95 (26) , 15264-15269.
    51. F. A. Wong, N. J. Anderson, S. J. Juzwin. Determination of a Synthetic Decapeptide in the Plasma of Monkeys and Rats by Narrowbore Highperformance Liquid Chromatography. Journal of Liquid Chromatography & Related Technologies 1998, 21 (7) , 1051-1062.
    52. MARIA PELLEGRINI, MIRIAM ROYO, MICHAEL CHOREV, DALE F. MIERKE. Conformational consequences of i, i + 3 cystine linkages: nucleation for α‐helicity?. The Journal of Peptide Research 1997, 49 (5) , 404-414.
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    55. Jean Rivier, Catherine Rivier, Steve Sutton, Antonio Miranda, Steven C. Koerber, Jozsef Gulyas, Sabine L. Lahrichi, Anne Corrigan, A. Grey Craig, Wylie Vale. Structure activity relationships (SAR) of corticotropin releasing factor. 1995, 195-198.
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    57. A. Miranda, S. Lahrichi, J. Gulyas, C. Rivier, S. Koerber, C. Miller, A. Corrigan, S. Sutton, A. Craig, W. Vale, J. Rivier. Competitive antagonists of the corticotropin releasing factor (CRF) scanned with a i-(i+3) Glu Lys Bridge. , 737-738.

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