Potential antileukemic and immunosuppressive drugs. Preparation and in vitro pharmacological activity of some 2,1,3-benzoxadiazoles (benzofurazans) and their N-oxides (benzofuroxans)

P. B. Ghosh, and Michael W. Whitehouse

J. Med. Chem., 1968, 11 (2), pp 305–311

DOI: 10.1021/jm00308a027

Publication Date: March 1968

Cite this:J. Med. Chem. 11, 2, 305-311

Note: In lieu of an abstract, this is the article's first page.

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Article

Potential antileukemic and immunosuppressive drugs. Preparation and in vitro pharmacological activity of some 2,1,3-benzoxadiazoles (benzofurazans) and their N-oxides (benzofuroxans)

Design, Synthesis, and Characterization of N-Oxide-Containing Heterocycles with in Vivo Sterilizing Antitubercular Activity

Antitumor Platinum(II) Complexes Containing Platinum-Based Moieties of Present Platinum Drugs and Furoxan Groups as Nitric Oxide Donors: Synthesis, DNA Interaction, and Cytotoxicity

Furoxans (1,2,5-Oxadiazole-N-Oxides) as Novel NO Mimetic Neuroprotective and Procognitive Agents

Copper(II)-Mediated Oxidative Transformation of vic-Dioxime to Furoxan: Evidence for a Copper(II)-Dinitrosoalkene Intermediate

Arylethenylbenzofuroxan Derivatives as Drugs for Chagas Disease: Multigram Batch Synthesis using a Wittig−Boden Process

Nitric Oxide Donors: Chemical Activities and Biological Applications

Efficient Synthesis of a Fluorescent Farnesylated Ras Peptide

1,2,5-Oxadiazole N-Oxide Derivatives and Related Compounds as Potential Antitrypanosomal Drugs: Structure−Activity Relationships

Rationalizing the Regioselectivity in Polynitroarene Anionic .sigma.-Adduct Formation. Relevance to Nucleophilic Aromatic Substitution

Rate and equilibrium studies in Jackson-Meisenheimer complexes

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Potential antileukemic and immunosuppressive drugs. Preparation and in vitro pharmacological activity of some 2,1,3-benzoxadiazoles (benzofurazans) and their N-oxides (benzofuroxans)

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